Salamah Maryana; Sipos Bence; Schelz Zsuzsanna; Zupkó István; Kiricsi Ágnes; Szalenko-Tőkés Ágnes; Rovó László; Katona Gábor; Balogh György Tibor; Pannonhalminé Csóka Ildikó:
Development, in vitro and ex vivo characterization of lamotrigine-loaded bovine serum albumin nanoparticles using QbD approach.
DRUG DELIVERY : JOURNAL OF DELIVERY AND TARGETING OF THERAPEUTIC AGENTS, 32 (1).
ISSN 1071-7544
(2025)
Khdar Zein Alabdeen; Le Minh Tam; Schelz Zsuzsanna; Zupkó István; Szakonyi Zsolt:
Aminodiols, aminotetraols and 1,2,3-triazoles based on allo-gibberic acid: stereoselective syntheses and antiproliferative activities.
RSC ADVANCES, 14 (49).
pp. 36698-36712.
ISSN 2046-2069
(2024)
Dembo António; Ferenczi Etelka; Jernei Tamás; Bor Andrea; Schelz Zsuzsanna; Zupkó István; Varga Szilárd; Csámpai Antal:
CuAAC-Based Synthesis, Copper-Catalyzed Aldehyde-Forming Hydrolytic Fission and Antiproliferative Evaluation of Novel Ferrocenoylamino-Substituted Triazole-Tethered Quinine–Chalcone Hybrids.
MOLECULES, 29 (2).
ISSN 1420-3049
(2024)
Gáborová Mária; Vágvölgyi Máté; Tayeb Bizhar Ahmed; Minorics Renáta; Zupkó István; Jurček Ondřej; Béni Szabolcs; Kubínová Renata; Balogh György Tibor; Hunyadi Attila:
Diterpenes Isolated from Three Different Plectranthus Sensu Lato Species and Their Antiproliferative Activities against Gynecological and Glioblastoma Cancer Cells.
ACS OMEGA, 9 (16).
pp. 18495-18504.
ISSN 2470-1343
(2024)
Keglevich Péter; Zupkó István; Szente Lajos; Puskás István; Szigetvári Áron; Mayer Szabolcs; Hazai László:
Does Vinblastine Retain its Anticancer Effect in the Presence of Cyclodextrin? A Preliminary Study.
PERIODICA POLYTECHNICA-CHEMICAL ENGINEERING, 68 (2).
pp. 133-139.
ISSN 0324-5853
(2024)
Szemerédi Nikoletta; Schelz Zsuzsanna; Horváth Dária Antónia; Rácz Bálint; Szatmári András G.; Muddather Hiba F.; Bózsity Noémi; Zupkó István; Spengler Gabriella:
Impact of V9302, a Competitive Antagonist of Transmembrane Glutamine Flux on Reversal of Resistance in Breast Cancer Cell Lines.
PHARMACEUTICS, 16 (7).
ISSN 1999-4923
(2024)
Szilvásy Nóra; Lajer Panna; Horváth Attila; Veres Katalin; Hohmann Judit; Schelz Zsuzsanna; Minorics Renáta; Zupkó István; Gáborik Zsuzsanna; Kis Emese; Temesszentandrási-Ambrus Csilla:
Modulation of Multispecific Transporters by Uncaria tomentosa Extract and Its Major Phytoconstituents.
PHARMACEUTICS, 16 (11).
ISSN 1999-4923
(2024)
Saidu Muhammad Bello; Krstić Gordana; Bombicz Petra; De Sourav; Barta Anita; Ali Hazhmat; Zupkó István; Berkecz Róbert; Gallah Umar Shehu; Rédei Dóra; Hohmann Judit:
New Members of the Centrapalus Coumarin and Pauciflorin Series from Centrapalus pauciflorus.
PHARMACEUTICS, 16 (7).
ISSN 1999-4923
(2024)
Fási Laura; Gonda Tímea; Crul-Tóth Noémi; Vass Máté; Gyovai András; Nagy Viktória; Ocsovszki Imre; Zupkó István; Kúsz Norbert; Nové Márta; Spengler Gabriella; Berkecz Róbert; Wang Hui-Chun; Chang Fang-Rong; Hunyadi Attila:
Preparation of dearomatized p‐coumaric acid derivatives as DNA damage response inhibitors with potent in vitro antitumor effect.
CHEMMEDCHEM, 19 (19).
ISSN 1860-7179
(2024)
Khdar Zein Alabdeen; Le Minh Tam; Schelz Zsuzsanna; Zupkó István; Szakonyi Zsolt:
Stereoselective synthesis and antiproliferative activity of allo-gibberic acid-based 1,3-aminoalcohols regioisomers.
RSC MEDICINAL CHEMISTRY, 15 (3).
pp. 874-887.
ISSN 2632-8682
(2024)
Ozsvár Dániel; Bózsity Noémi; Zupkó István; Szakonyi Zsolt:
Synthesis and Study of the Structure–Activity Relationship of Antiproliferative N-Substituted Isosteviol-Based 1,3-Aminoalcohols.
PHARMACEUTICALS, 17 (2).
ISSN 1424-8247
(2024)
Le Minh Tam; Njangiru Isaac Kinyua; Vincze Anna; Zupkó István; Balogh György Tibor; Szakonyi Zsolt:
Synthesis and medicinal chemical characterisation of antiproliferative O,N-functionalised isopulegol derivatives.
RSC ADVANCES, 14 (26).
pp. 18508-18518.
ISSN 2046-2069
(2024)
Bózsity-Faragó Noémi; Nagy Viktória; Szabó Johanna; Pálházi Balázs; Kele Zoltán; Resch Vivien; Paragi Gábor; Zupkó István; Minorics Renáta; Mernyák Erzsébet:
Synthesis of Estrone Heterodimers and Evaluation of Their In Vitro Antiproliferative Activity.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 25 (8).
ISSN 1661-6596
(2024)
Kusuma Ikhwan Yuda; Abdallah Hiba Faroug Muddather; Kurnianto Arie Arizandi; Bahar Muhammad Akbar; Kurniasih Khamdiyah Indah; Tololiu Kevin Efrain; Schelz Zsuzsanna; Zupkó István; Matuz Mária; Benkő Ria:
Telepharmacy in Indonesia: Navigating Knowledge, Perception, and Readiness Among 6,000 Pharmacists and Related Sociodemographic Determinants.
TELEMEDICINE AND E-HEALTH, 30 (9).
pp. 2483-2494.
ISSN 1530-5627
(2024)
Ahmed Sara Hassan Hassan; Tayeb Bizhar Ahmed; Gonda Tímea; Girst Gábor; Szőri Kornél; Berkecz Róbert; Zupkó István; Minorics Renáta; Hunyadi Attila:
Thymoquinone-protoflavone hybrid molecules as potential antitumor agents.
PLOS ONE, 19 (1).
ISSN 1932-6203
(2024)
Said Awad I.; Gajdács Márió; Zupkó István; Haukka Matti; Palkó Márta:
Angular Regioselective Synthesis of Varied Functionalized Hexahydro-1,2,4-triazolo[4,3-a]quinazolin-9-ones and Their Antiproliferative Action.
MOLECULES, 28 (9).
ISSN 1420-3049
(2023)
Krstić Gordana; Saidu Muhammad Bello; Barta Anita; Vágvölgyi Máté; Ali Hazhmat; Zupkó István; Berkecz Róbert; Gallah Umar Shehu; Rédei Dóra; Hohmann Judit:
Anticancer Meroterpenoids from Centrapalus pauciflorus leaves: Chromone- and 2,4-Chromadione-Monoterpene Derivatives.
ACS OMEGA, 8 (34).
pp. 31389-31398.
ISSN 2470-1343
(2023)
Senobar Tahaei Seyyed Ashkan; Kulmány Ágnes; Minorics Renáta; Kiss Anita; Szabó Zoltán; Germán Péter; Szebeni Gábor; Gémes Nikolett; Mernyák Erzsébet; Zupkó István:
Antiproliferative and Antimetastatic Properties of 16-Azidomethyl Substituted 3-O-Benzyl Estrone Analogs.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 24 (18).
ISSN 1661-6596
(2023)
Nagy Viktória; Mounir Raji; Szebeni Gábor J.; Szakonyi Zsolt; Gémes Nikolett; Minorics Renáta; Germán Péter; Zupkó István:
Investigation of Anticancer Properties of Monoterpene-Aminopyrimidine Hybrids on A2780 Ovarian Cancer Cells.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 24 (13).
ISSN 1661-6596
(2023)
Kovács Tibor; Lajter Ildikó; Kúsz Norbert; Schelz Zsuzsanna; Bózsity-Faragó Noémi; Borbás Anikó; Zupkó István; Krupitza Georg; Frisch Richard; Hohmann Judit; Vasas Andrea; Mándi Attila:
Isolation and NMR Scaling Factors for the Structure Determination of Lobatolide H, a Flexible Sesquiterpene from Neurolaena lobata.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 24 (6).
ISSN 1661-6596
(2023)
Ferencz Elek; Spengler Gabriella; Zupkó István; Vollár Martin; Zomborszki Zoltán Péter; Kúsz Norbert; Hohmann Judit; Kovács Balázs; Csupor Dezső; Laczkó-Zöld Eszter; Csupor-Löffler Boglárka:
Isolation of compounds from the roots of Ambrosia artemisiifolia and their effects on human cancer cell lines.
ZEITSCHRIFT FÜR NATURFORSCHUNG C-A JOURNAL OF BIOSCIENCES, 78 (7-8).
pp. 299-305.
ISSN 0939-5075
(2023)
Lőrincz Eszter Boglárka; Tóth Gergely; Spolárics Júlia; Herczeg Mihály; Hodek Jan; Zupkó István; Minorics Renáta; Ádám Dorottya; Oláh Attila; Zouboulis Christos C.; Weber Jan; Nagy Lajos; Ostorházi Eszter; Bácskay Ildikó; Borbás Anikó; Herczegh Pál; Bakai-Bereczki Ilona:
Mannich-type modifications of (−)-cannabidiol and (−)-cannabigerol leading to new, bioactive derivatives.
SCIENTIFIC REPORTS, 13 (1).
ISSN 2045-2322
(2023)
Saidu Muhammad Bello; Krstić Gordana; Todorović Nina; Berkecz Róbert; Ali Hazhmat; Zupkó István; Hohmann Judit; Rédei Dóra:
Monoterpenoid 5-methylcoumarins from Centrapalus pauciflorus with antiproliferative activity.
ARABIAN JOURNAL OF CHEMISTRY, 16 (6).
ISSN 1878-5352
(2023)
Krstić Gordana; Saidu Muhammad Bello; Bombicz Petra; De Sourav; Ali Hazhmat; Zupkó István; Berkecz Róbert; Gallah Umar Shehu; Rédei Dóra; Hohmann Judit:
Pauciflorins A–E, Unexpected Chromone–Monoterpene-Derived Meroterpenoids from Centrapalus pauciflorus.
JOURNAL OF NATURAL PRODUCTS, 86 (4).
pp. 891-896.
ISSN 0163-3864
(2023)
Bai Dorottya; Schelz Zsuzsanna; Erdős Dóra; Kis Anna K.; Nagy Viktória; Zupkó István; Balogh György Tibor; Szakonyi Zsolt:
Stereoselective Synthesis and Antiproliferative Activities of Tetrafunctional Diterpene Steviol Derivatives.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 24 (2).
ISSN 1661-6596
(2023)
Bai Dorottya; Schelz Zsuzsanna; Boncz Mária Fanni; Zupkó István; Szakonyi Zsolt:
Stereoselective Synthesis and Antiproliferative Activity of Steviol-Based Diterpene 1,3-Aminoalcohol Regioisomers.
MOLECULES, 28 (24).
ISSN 1420-3049
(2023)
Kovács Édua; Ali Hazhmat; Minorics Renáta; Traj Péter; Resch Vivien Erzsébet; Paragi Gábor; Bruszel Bella; Zupkó István; Mernyák Erzsébet:
Synthesis and Antiproliferative Activity of Steroidal Diaryl Ethers.
MOLECULES, 28 (3).
ISSN 1420-3049
(2023)
Németh-Rieder Alexandra; Keglevich Péter; Hunyadi Attila; Latif Ahmed Dhahir; Zupkó István; Hazai László:
Synthesis and In Vitro Anticancer Evaluation of Flavone—1,2,3-Triazole Hybrids.
MOLECULES, 28 (2).
ISSN 1420-3049
(2023)
Bamou Zahra Fatima; Le Minh Tam; Tayeb Bizhar Ahmed; Tahaei Seyyed Ashkan Senobar; Minorics Renáta; Zupkó István; Szakonyi Zsolt:
Antiproliferative Activity of (-)-Isopulegol-based 1,3-Oxazine, 1,3-Thiazine and 2,4-Diaminopyrimidine Derivative.
CHEMISTRYOPEN, 11 (10).
ISSN 2191-1363
(2022)
Katona Gábor; Sabir Fakhara; Sipos Bence; Naveed Muhammad; Schelz Zsuzsanna; Zupkó István; Pannonhalminé Csóka Ildikó:
Development of Lomustine and n-Propyl Gallate Co-Encapsulated Liposomes for Targeting Glioblastoma Multiforme via Intranasal Administration.
PHARMACEUTICS, 14 (3).
Terjedelem: 22-Azonosító: 631.
ISSN 1999-4923
(2022)
Mounir Raji; Le Minh Tam; Huynh Thu; Szekeres András; Nagy Viktória; Zupkó István; Szakonyi Zsolt:
Divergent Synthesis, Antiproliferative and Antimicrobial Studies of 1,3‐Aminoalcohol and 3‐Amino‐1,2‐Diol Based Diaminopyrimidines.
CHEMISTRY & BIODIVERSITY, 19 (5).
Terjedelem: 11-Azonosító: e202200077.
ISSN 1612-1872
(2022)
Kata Diána; Gróf Ilona; Hoyk Zsófia; Ducza Eszter; Deli Mária Anna; Zupkó István; Földesi Imre:
Immunofluorescent Evidence for Nuclear Localization of Aromatase in Astrocytes in the Rat Central Nervous System.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 23 (16).
Terjedelem: 21 p.-Azonosító: 8946.
ISSN 1661-6596
(2022)
Dávid Csilla Zsuzsanna; Kúsz Norbert; Pinke Gyula; Kulmány Ágnes Erika; Zupkó István; Hohmann Judit; Vasas Andrea:
Jacaranone Derivatives with Antiproliferative Activity from Crepis pulchra and Relevance of This Group of Plant Metabolites.
PLANTS-BASEL, 11 (6).
Terjedelem: 11-Azonosító: 782.
ISSN 2223-7747
(2022)
Sipos Bence; Pannonhalminé Csóka Ildikó; Szivacski Nimród; Budai-Szűcs Mária; Schelz Zsuzsanna; Zupkó István; Révész Piroska; Volk Balázs; Katona Gábor:
Mucoadhesive meloxicam-loaded nanoemulsions: development, characterization and nasal applicability studies.
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 175.
Terjedelem: 10-Azonosító: 106229.
ISSN 0928-0987
(2022)
Molnár Barnabás; Njangiru Isaac Kinyua; Mótyán Gergő; Leits Péter; Zupkó István; Minorics Renáta; Balogh György Tibor; Nagyné Frank Éva:
Regioselective synthesis, physicochemical properties and anticancer activity of 2-aminomethylated estrone derivatives.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 219.
Terjedelem: 13 p-Azonosító: 106064.
ISSN 0960-0760
(2022)
Sipos Bence; Pannonhalminé Csóka Ildikó; Ambrus Rita; Schelz Zsuzsanna; Zupkó István; Balogh György Tibor; Katona Gábor:
Spray-dried indomethacin-loaded polymeric micelles for the improvement of intestinal drug release and permeability.
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 174.
Terjedelem: 11-Azonosító: 106200.
ISSN 0928-0987
(2022)
Khdar Zein Alabdeen; Le Minh Tam; Schelz Zsuzsanna; Zupkó István; Szakonyi Zsolt:
Stereoselective Synthesis and Application of Gibberellic Acid-Derived Aminodiols.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 23 (18).
Terjedelem: 24 p.-Azonosító: 10366.
ISSN 1661-6596
(2022)
Mounir Raji; Le Minh Tam; Csámpai Antal; Nagy Viktória; Zupkó István; Szakonyi Zsolt:
Stereoselective Synthesis and Applications of Pinane-Based Chiral 1,4-Amino Alcohol Derivatives.
SYNTHESIS-STUTTGART, 54 (17).
pp. 3831-3844.
ISSN 0039-7881
(2022)
Ristovski Jovana; Minorics Renáta; Bartha Sándor; Jankovic Nenad; Zupkó István:
The evaluation of the anticancer activity of the Biginelli hybrids and pharmacokinetic profiling based on their retention parameters.
Journal of Molecular Structure, 1254.
Terjedelem: 12-Azonosító: 132373.
ISSN 0022-2860
(2022)
Kulmány Ágnes Erika; Nagyné Frank Éva; Kovács Dóra; Kirisits Kerstin; Krupitza Georg; Neuperger Patricia; Alföldi Róbert; Puskás László; Szebeni Gábor; Zupkó István:
Antiproliferative and antimetastatic characterization of an exo-heterocyclic androstane derivative against human breast cancer cell lines.
BIOMEDICINE & PHARMACOTHERAPY, 140.
Terjedelem: 17 p-Azonosító: 111728.
ISSN 0753-3322
(2021)
Balogh Nikoletta; Schelz Zsuzsanna; Zupkó István:
Az emlődaganatok farmakoterápiás lehetőségei.
GYÓGYSZERÉSZET, 65.
pp. 93-99.
ISSN 0017-6036
(2021)
Kulmány Ágnes Erika; Nagyné Frank Éva; Papp Dóra Anna; Szekeres András; Szebeni Gábor; Zupkó István:
Biological Evaluation of Antiproliferative and Anti-Invasive Properties of an Androstadiene Derivative on Human Cervical Cancer Cell Lines.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 214.
Terjedelem: 12 p-Azonosító: 105990.
ISSN 0960-0760
(2021)
Danciu Corina; Cioanca Oana; Watz Farcaș Claudia; Hancianu Monica; Racoviceanu Roxana; Muntean Delia; Zupkó István; Oprean Camelia; Tatu Calin; Paunescu Virgil; Proks Maria; Diaconeasa Zorita; Soica Codruta; Pinzaru Iulia; Dehelean Cristina:
Botanical Therapeutics (Part II): Antimicrobial and In Vitro Anticancer Activity against MCF7 Human Breast Cancer Cells of Chamomile, Parsley and Celery Alcoholic Extracts.
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, 21 (2).
pp. 187-200.
ISSN 1871-5206
(2021)
Gospodinova Zlatina I.; Zupkó István; Bózsity Noémi; Manova Vasilissa I.; Georgieva Mariyana S.; Todinova Svetla J.; Taneva Stefka Germanova; Krasteva Maria Emileva; Ocsovszki Imre:
Cotinus coggygria Scop. induces cell cycle arrest, apoptosis, genotoxic effects, thermodynamic and epigenetic events in MCF7 breast cancer cells.
ZEITSCHRIFT FÜR NATURFORSCHUNG C-A JOURNAL OF BIOSCIENCES, 76 (3-4).
pp. 129-140.
ISSN 0939-5075
(2021)
Kulmány Ágnes Erika; Herman Bianka Edina; Zupkó István; Sinreih Masa; Rižner Tea Lanišnik; Savić Marina; Oklješa Aleksandar; Nikolić Andrea; Nagy Viktória; Ocsovszki Imre; Szécsi Mihály; Jovanovic-Santa Suzana:
Heterocyclic androstane and estrane D-ring modified steroids : microwave-assisted synthesis, steroid-converting enzyme inhibition, apoptosis induction, and effects on genes encoding estrogen inactivating enzymes.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 214.
Terjedelem: 13 p-Azonosító: 105997.
ISSN 0960-0760
(2021)
Vasas Andrea; Lajter Ildikó; Kúsz Norbert; Király Sándor Balázs; Kovács Tibor; Kurtán Tibor; Bózsity Noémi; Nagy Nikolett; Schelz Zsuzsanna; Zupkó István; Krupitza Georg; Frisch Richard; Mándi Attila; Hohmann Judit:
Isolation, Structure Determination of Sesquiterpenes from Neurolaena lobata and Their Antiproliferative, Cell Cycle Arrest-Inducing and Anti-Invasive Properties against Human Cervical Tumor Cells.
PHARMACEUTICS, 13 (12).
Terjedelem: 25 p-Azonosító: 2088.
ISSN 1999-4923
(2021)
Mernyák Erzsébet; Bartha Sándor; Kóczán Lili; Jójárt Rebeka; Resch Vivien; Paragi Gábor; Vágvölgyi Máté; Hunyadi Attila; Bruszel Bella; Zupkó István; Minorics Renáta:
Microwave-assisted Phospha-Michael addition reactions in the 13 alpha-oestrone series and in vitro antiproliferative properties.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 36 (1).
pp. 1931-1937.
ISSN 1475-6366
(2021)
Kiss Anita; Jójárt Rebeka; Mernyák Erzsébet; Bartha Sándor; Minorics Renáta; Zupkó István; Schneider Gyula:
Novel preparation of substituted oxazolines condensed to d-ring of estrane skeleton and characterization of their antiproliferative properties.
STEROIDS, 176.
Terjedelem: 6 p-Azonosító: 108911.
ISSN 0039-128X
(2021)
Kryczyk-Poprawa Agata; Zupkó István; Bérdi Péter; Żmudzki Paweł; Piotrowska Joanna; Pękala Elżbieta; Berdys Aleksandra; Muszyńska Bożena; Opoka Włodzimierz:
Photodegradation of Bexarotene and Its Implication for Cytotoxicity.
PHARMACEUTICS, 13 (8).
Terjedelem: 18 p-Azonosító: 1220.
ISSN 1999-4923
(2021)
Ozsvár Dániel; Nagy Viktória; Zupkó István; Szakonyi Zsolt:
Synthesis and Biological Application of Isosteviol-Based 1,3-Aminoalcohols.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 22 (20).
Terjedelem: 20-Azonosító: 11232.
ISSN 1661-6596
(2021)
Mohamed El Haimer; Palkó Márta; Matti Haukka; Gajdács Márió; Zupkó István; Fülöp Ferenc:
Synthesis and biological evaluation of the new ring system benzo[f]pyrimido[1,2-d][1,2,3]triazolo[1,5-a][1,4]diazepine and its cycloalkane and cycloalkene condensed analogues.
RSC ADVANCES, 11 (12).
pp. 6952-6957.
ISSN 2046-2069
(2021)
Jójárt Rebeka; Senobar Tahaei Seyyed Ashkan; Trungel-Nagy Péter; Kele Zoltán; Minorics Renáta; Paragi Gábor; Zupkó István; Mernyák Erzsébet:
Synthesis and evaluation of anticancer activities of 2- or 4-substituted 3-(N-benzyltriazolylmethyl)-13α-oestrone derivatives.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 36 (1).
pp. 58-67.
ISSN 1475-6366
(2021)
El Haimer Mohamed; Faragó Tünde; Schelz Zsuzsanna; Zupkó István; Palkó Márta:
Synthesis of Alicyclic 2-Methylenethiazolo[2,3-b]quinazolinone Derivatives via Base-Promoted Cascade Reactions.
SYNTHESIS-STUTTGART, 53 (Suppl.).
A-H.
ISSN 0039-7881
(2021)
Traj Péter; Ali Hazhmat; Németh Anett; Dajcs Sámuel Trisztán; Tömösi Ferenc; Lanisnik-Rizner Tea; Zupkó István; Mernyák Erzsébet:
Transition metal-catalyzed A-ring C–H activations and C(sp2)–C(sp2) couplings in the 13α-estrone series and in vitro evaluation of antiproliferative properties.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 36 (1).
pp. 895-902.
ISSN 1475-6366
(2021)
Fási Laura; Latif Ahmed Dhahir; Zupkó István; Lévai Sándor; Dékány Miklós; Béni Zoltán; Könczöl Árpád; Balogh György Tibor; Hunyadi Attila:
AAPH or Peroxynitrite-Induced Biorelevant Oxidation of Methyl Caffeate Yields a Potent Antitumor Metabolite.
BIOMOLECULES, 10 (11).
Azonosító: 1537-Terjedelem: 13 p.
ISSN 2218-273X
(2020)
Csupor Dezső; Kurtán Tibor; Vollár Martin; Kúsz Norbert; E Kövér Katalin; Mándi Attila; Szűcs Péter; Marschall Marianna; Tahaei Seyyed A. Senobar; Zupkó István; Hohmann Judit:
Correction to Pigments of the Moss Paraleucobryum longifolium: Isolation and Structure Elucidation of Prenyl-Substituted 8,8′-Linked 9,10-Phenanthrenequinone Dimers.
JOURNAL OF NATURAL PRODUCTS, 83 (4).
p. 1355.
ISSN 0163-3864
(2020)
Hajdú Zsuzsanna; Forgó Péter; Király Gergely; Pinke Gyula; Zupkó István; Hohmann Judit:
Isolation Of Chemical Constituents From Filago Vulgaris And Antiproliferative Activity Of The Plantextract And Its Flavonoid Against Human Tumor Cell Lines.
PAKISTAN JOURNAL OF PHARMACEUTICAL SCIENCES, 33 (4).
pp. 1593-1597.
ISSN 1011-601X
(2020)
Bús Csaba; Kulmány Ágnes Erika; Kúsz Norbert; Gonda Tímea; Zupkó István; Mándi Attila; Kurtán Tibor; Tóth Barbara; Hohmann Judit; Hunyadi Attila; Vasas Andrea:
Oxidized Juncuenin B Analogues with Increased Antiproliferative Activity on Human Adherent Cell Lines: Semisynthesis and Biological Evaluation.
JOURNAL OF NATURAL PRODUCTS, 83 (11).
pp. 3250-3261.
ISSN 0163-3864
(2020)
Jójárt Rebeka; Ali Hazhmat; Horváth Gergely; Kele Zoltán; Zupkó István; Mernyák Erzsébet:
Pd-Catalyzed Suzuki–Miyaura couplings and evaluation of 13α-estrone derivatives as potential anticancer agents.
STEROIDS, 164.
Terjedelem: 10 p.-Azonosító: 108731.
ISSN 0039-128X
(2020)
Kryczyk-Poprawa Agata; Zupkó István; Bérdi Péter; Żmudzki Paweł; Popiół Justyna; Muszyńska Bożena; Opoka Włodzimierz:
Photostability Testing of a Third-Generation Retinoid—Tazarotene in the Presence of UV Absorbers.
PHARMACEUTICS, 12 (9).
Terjedelem: 20 p.-Azonosító: 899.
ISSN 1999-4923
(2020)
Csupor Dezső; Kurtán Tibor; Vollár Martin; Kúsz Norbert; Kövér Katalin E.; Mándi Attila; Szűcs Péter; Marschall Marianna; Senobar Tahaei Seyyed Ashkan; Zupkó István; Hohmann Judit:
Pigments of the Moss Paraleucobryum longifolium: Isolation and Structure Elucidation of Prenyl-Substituted 8,8′-Linked 9,10-Phenanthrenequinone Dimers.
JOURNAL OF NATURAL PRODUCTS, 83 (2).
pp. 268-276.
ISSN 0163-3864
(2020)
Latif Ahmed Dhahir; Jernei Tamás; Podolski-Renić Ana; Kuo Ching-Ying; Vágvölgyi Máté; Girst Gábor; Zupkó István; Develi Sedef; Ulukaya Engin; Wang Hui-Chun; Pešić Milica; Csámpai Antal; Hunyadi Attila:
Protoflavone-Chalcone Hybrids Exhibit Enhanced Antitumor Action through Modulating Redox Balance, Depolarizing the Mitochondrial Membrane, and Inhibiting ATR-Dependent Signaling.
ANTIOXIDANTS, 9 (6).
Azonosító: 519-Terjedelem: 18 p.
ISSN 2076-3921
(2020)
Vágvölgyi Máté; Bélteky Péter; Bogdán Dóra; Nové Márta; Spengler Gabriella; Latif Ahmed Dhahir; Zupkó István; Gáti Tamás; Tóth Gábor; Kónya Zoltán; Hunyadi Attila:
Squalenoylated Nanoparticle Pro-Drugs of Adjuvant Antitumor 11α-Hydroxyecdysteroid 2,3-Acetonides Act as Cytoprotective Agents Against Doxorubicin and Paclitaxel.
FRONTIERS IN PHARMACOLOGY, 11.
Azonosító: 552088-Terjedelem: 14 p.
ISSN 1663-9812
(2020)
Ozsvár Dániel; Nagy Viktória; Zupkó István; Szakonyi Zsolt:
Stereoselective Synthesis and Antiproliferative Activity of Steviol-Based Diterpen Aminodiols.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 21 (1).
Azonosító: 184-Terjedelem: 17 p.
ISSN 1661-6596
(2020)
Kuskucu K.; Akyildiz V.; Kulmány Á.; Ergün Y.; Zencir S.; Zupkó István; Durdagi S.; Zaka M.; Sahin K.; Orhan H.; Topcu Z.:
Structural modification of ellipticine derivatives with alkyl groups of varying length is influential on their effects on human DNA topoisomerase II: a combined experimental and computational study.
MEDICINAL CHEMISTRY RESEARCH, 29.
pp. 189-198.
ISSN 1054-2523
(2020)
Keglevich András; Dányi Leonetta; Rieder Alexandra; Horváth Dorottya; Szigetvári Áron; Dékány Miklós; Szántay Csaba, ifj.; Latif Ahmed Dhahir; Hunyadi Attila; Zupkó István; Keglevich Péter; Hazai László:
Synthesis and Cytotoxic Activity of New Vindoline Derivatives Coupled to Natural and Synthetic Pharmacophores.
MOLECULES, 25 (4).
Azonosító: 1010-Terjedelem: 19 p.
ISSN 1420-3049
(2020)
Minda Daliana; Avram Stefana; Pavel Ioana Zinuca; Kis Brigitta; Ghitu Alexandra; Zupkó István; Dehelean Cristina; Buda Valentina; Diaconeasa Zorita; Scurtu Alexandra; Vlad Alexa; Danicu Corina:
An in vitro Evaluation of Apigenin and Apigenin-7-O-glucoside Against HeLa Human Cervical Cancer Cell Line.
REVISTA DE CHIMIE, 71 (2).
pp. 140-144.
ISSN 0034-7752
(2020)
Szabó Renáta; Börzsei Denise; Szabó Zsuzsanna; Nagyné Hoffmann Alexandra; Zupkó István; Priksz Dániel; Kupai Krisztina; Varga Csaba; Pósa Anikó:
A potential involvement of anandamide in the modulation of HO/NOS systems: Women, menopause, and “medical cannabinoids”.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 21 (22).
Terjedelem: 13-Azonosító: 8801.
ISSN 1661-6596
(2020)
Mótyán Gergő; Gopisetty Mohana Krishna; Zupkó István; Zupkó István; Zupkó István; Nagyné Frank Éva; Csontné Kiricsi Mónika:
Anti-Cancer Activity of Novel Dihydrotestosterone-Derived Ring A-Condensed Pyrazoles on Androgen Non-Responsive Prostate Cancer Cell Lines.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 20 (9).
Azonosító: 2170-Terjedelem: 20 p.
ISSN 1661-6596
(2019)
Gajdács Márió; Zupkó István:
Az antibiotikum rezisztencia krízis: lépést tudnak-e tartani a gyógyszerfejlesztő cégek?
GYÓGYSZERÉSZET, 63 (12).
pp. 736-742.
ISSN 0017-6036
(2019)
Tóth Ildikó; Nyergesné Illés Erzsébet; Szekeres Márta; Zupkó István; Turcu Rodica; Tombácz Etelka:
Chondroitin-Sulfate-A-Coated Magnetite Nanoparticles: Synthesis, Characterization and Testing to Predict Their Colloidal Behavior in Biological Milieu.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 20 (17).
Terjedelem: 19 p-Azonosító: 4096.
ISSN 1661-6596
(2019)
Nicolov Mirela; Ghiulai Roxana M.; Voicu Mirela; Mioc Marius; Duse Adina Octavia; Roman Roxana; Ambrus Rita; Zupkó István; Moaca Elena Alina; Coricovac Dorina E.; Farcas Claudia; Racoviceanu Roxana Marcela; Danciu Corina; Dehelean Cristina-Adriana; Soica Codruta:
Cocrystal Formation of Betulinic Acid and Ascorbic Acid: Synthesis, Physico-Chemical Assessment, Antioxidant, and Antiproliferative Activity.
Frontiers in Chemistry, 7.
Azonosoító: 92-Terjedelem: 11 p.
ISSN 2296-2646
(2019)
Ghițu Alexandra; Schwiebs Anja; Radeke Heinfried H.; Avram Ştefana; Zupkó István; Bor Andrea; Pavel Ioana Zinuca; Dehelean Cristina Adriana; Oprean Camelia; Bojin Florina; Farcas Claudia; Soica Codruta; Duicu Oana; Danciu Corina:
A Comprehensive Assessment of Apigenin as an Antiproliferative, Proapoptotic, Antiangiogenic and Immunomodulatory Phytocompound.
NUTRIENTS, 11 (4).
Paper 858-19 p.
ISSN 2072-6643
(2019)
Kiss Tivadar; Timár Zoltán; Szabó Andrea; Hebőkné Lukács Anita; Velky Viktória; Oszlánczi Gábor; Horváth Edina; Takács István; Zupkó István; Csupor Dezső:
Effect of green tea on the gastrointestinal absorption of amoxicillin in rats.
BMC PHARMACOLOGY & TOXICOLOGY, 20.
Terjedelem: 7 p-Azonosító: 54.
ISSN 2050-6511
(2019)
Kuo Ching-Ying; Schelz Zsuzsanna; Tóth Barbara; Vasas Andrea; Ocsovszki Imre; Chang Fang-Rong; Hohmann Judit; Zupkó István; Wang Hui-Chun:
Investigation of natural phenanthrenes and the antiproliferative potential of juncusol in cervical cancer cell lines.
PHYTOMEDICINE, 58.
Paper 152770-10 p.
ISSN 0944-7113
(2019)
Hammadi Reham; Kúsz Norbert; Mwangi Peter W.; Kulmány Ágnes Erika; Zupkó István; Orvos Péter; Tálosi László; Hohmann Judit; Vasas Andrea:
Isolation and Pharmacological Investigation of Compounds From Euphorbia matabelensis.
NATURAL PRODUCT COMMUNICATIONS, 14 (7).
ISSN 1934-578X
(2019)
Stefkó Dóra; Kúsz Norbert; Csorba Attila; Jakab Gusztáv; Bérdi Péter; Zupkó István; Hohmann Judit; Vasas Andrea:
Phenanthrenes from Juncus atratus with antiproliferative activity.
TETRAHEDRON, 75 (1).
pp. 116-120.
ISSN 0040-4020
(2019)
Danciu Corina; Muntean Delia; Alexa Ersilia; Farcas Claudia; Oprean Camelia; Zupkó István; Bor Andrea; Minda Daliana; Proks Maria; Buda Valentina; Hancianu Monica; Cioanca Oana; Soica Codruta; Popescu Sofia; Dehelean Cristina Adriana:
Phytochemical Characterization and Evaluation of the Antimicrobial, Antiproliferative and Pro-Apoptotic Potential of Ephedra alata Decne. Hydroalcoholic Extract against the MCF-7 Breast Cancer Cell Line.
MOLECULES, 24 (1).
Paper 13-15 p.
ISSN 1420-3049
(2019)
Tastan Pelin; Hajdú Zsuzsanna; Kúsz Norbert; Zupkó István; Sinka Izabella; Kivçak Bijen; Hohmann Judit:
Sesquiterpene Lactones and Flavonoids from Psephellus pyrrhoblepharus with Antiproliferative Activity on Human Gynecological Cancer Cell Lines.
MOLECULES, 24 (17).
Terjedelem: 9 p-Azonosító: 3165.
ISSN 1420-3049
(2019)
Kiss Anita; Wölfling János; Mernyák Erzsébet; Nagyné Frank Éva; Benke Zsanett Amália; Zupkó István; Schneider Gyula:
Stereocontrolled synthesis of the four possible 3-methoxy and 3-benzyloxy-16-triazolyl-methyl-estra-17-ol hybrids and their antiproliferative activities.
STEROIDS, 152.
Azonosító: 108500-Terjedelem: 14 p.
ISSN 0039-128X
(2019)
Kiss Anita; Wölfling János; Mernyák Erzsébet; Nagyné Frank Éva; Gyovai András; Kulmány Ágnes Erika; Zupkó István; Schneider Gyula:
Stereoselective Synthesis of New Type of Estradiol Hybrid Molecules and their Antiproliferative Activities.
STEROIDS, 148.
pp. 63-72.
ISSN 0039-128X
(2019)
Latif Ahmed Dhahir; Gonda Tímea; Vágvölgyi Máté; Kúsz Norbert; Kulmány Ágnes Erika; Ocsovszki Imre; Zomborszki Zoltán Péter; Zupkó István; Hunyadi Attila:
Synthesis and In Vitro Antitumor Activity of Naringenin Oxime and Oxime Ether Derivatives.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 20 (9).
Paper 2184-12 p.
ISSN 1661-6596
(2019)
Nowikow Christina; Fuerst Rita; Kauderer Maria; Dank Christian; Schmid Walther; Hajduch Marian; Rehulka Jiri; Gurska Sona; Mokshyna Olena; Polishchuk Pavel; Zupkó István; Dzubak Petr; Rinner Uwe:
Synthesis and biological evaluation of cis-restrained carbocyclic combretastatin A-4 analogs: Influence of the ring size and saturation on cytotoxic properties.
BIOORGANIC & MEDICINAL CHEMISTRY, 27 (19).
Terjedelem: 13 p-Azonosító: 115032.
ISSN 0968-0896
(2019)
Huber Imre; Zupkó István; Gyovai András; Horváth Péter; Kiss Eszter; Gulyás Gergely; Schmidt János; Perjési Pál:
A novel cluster of C5-curcuminoids: design, synthesis, in vitro antiproliferative activity and DNA binding of bis(arylidene)-4-cyclanone derivatives based on 4-hydroxycyclohexanone scaffold.
RESEARCH ON CHEMICAL INTERMEDIATES, 45 (9).
pp. 4711-4735.
ISSN 0922-6168
(2019)
Sinka Izabella; Kiss Anita; Mernyák Erzsébet; Wölfling János; Schneider Gyula; Ocsovszki Imre; Kuo Ching-Ying; Wang Hui-Chun; Zupkó István:
Antiproliferative and antimetastatic properties of 3-benzyloxy-6-hydroxymethylene-estradiol analogs against breast cancer cell lines.
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 123.
pp. 362-370.
ISSN 0928-0987
(2018)
Vollár Martin; Gyovai András; Szűcs Péter; Zupkó István; Marschall Marianna; Csupor-Löffler Boglárka; Bérdi Péter; Vecsernyés Anikó; Csorba Attila; Liktor-Busa Erika; Zsoldiné Urbán Edit; Csupor Dezső:
Antiproliferative and antimicrobial activities of selected bryophytes.
MOLECULES, 23 (7).
Terjedelem: 15 p.-Azonosító: 1520.
ISSN 1420-3049
(2018)
Danciu Corina; Pinzaru Iulia Andreea; Dehelean Cristina Adriana; Hancianu Monica; Zupkó István; Navolan Dan; Licker Monica; Ghiulai Roxana Maria; Şoica Codruta Marinela:
Antiproliferative and antimicrobial properties of pure and encapsulated rutin.
FARMACIA (BUCHAREST), 66 (2).
pp. 302-308.
ISSN 0014-8237
(2018)
Gyovai András; Minorics Renáta; Kiss Anita; Mernyák Erzsébet; Schneider Gyula; Szekeres András; Kerekes Erika Beáta; Ocsovszki Imre; Zupkó István:
Antiproliferative properties of newly synthesized 19-nortestosterone analogs without substantial androgenic activity.
FRONTIERS IN PHARMACOLOGY, 9.
Terjedelem: 11 p.-Azonosító: 825.
ISSN 1663-9812
(2018)
Rédei Dóra; Kúsz Norbert; Jedlinszki Nikoletta; Blazsó Gábor; Zupkó István; Hohmann Judit:
Bioactivity-Guided Investigation of the Anti-Inflammatory Activity of Hippophae rhamnoides Fruits.
PLANTA MEDICA: NATURAL PRODUCTS AND MEDICINAL PLANT RESEARCH, 84.
pp. 26-33.
ISSN 0032-0943
(2018)
Danciu Corina; Zupkó István; Bor Andrea; Schwiebs Anja; Radeke Heinfried; Hancianu Monica; Cioanca Oana; Alexa Ersilia; Oprean Camelia; Bojin Florina; Soica Codruta; Paunescu Virgil; Dehelean Cristina Adriana:
Botanical Therapeutics: Phytochemical Screening and Biological Assessment of Chamomile, Parsley and Celery Extracts against A375 Human Melanoma and Dendritic Cells.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 19 (11).
Paper 3624-20 p.
ISSN 1661-6596
(2018)
Vlaisavljević Sanja; Šibul Filip; Sinka Izabella; Zupkó István; Ocsovszki Imre; Jovanovic-Santa Suzana:
Chemical composition, antioxidant and anticancer activity of licorice from
Fruska Gora locality.
INDUSTRIAL CROPS AND PRODUCTS, 112.
pp. 217-224.
ISSN 0926-6690
(2018)
Kovács Bernadett; Béni Zoltán; Dékány Miklós; Bózsity Noémi; Zupkó István; Hohmann Judit; Ványolós Attila:
Isolation and structure determination of antiproliferative secondary metabolites from the potato earthball mushroom, Scleroderma bovista (Agaricomycetes).
INTERNATIONAL JOURNAL OF MEDICINAL MUSHROOMS, 20 (5).
pp. 411-418.
ISSN 1521-9437
(2018)
Nyergesné Illés Erzsébet; Szekeres Márta; Tóth Ildikó; Szabó Ákos; Iván Béla; Turcu Rodica; Vékás Ladislau; Zupkó István; Jaics György; Csákiné Tombácz Etelka:
Multifunctional PEG-carboxylate copolymer coated superparamagnetic iron oxide nanoparticles for biomedical application.
JOURNAL OF MAGNETISM AND MAGNETIC MATERIALS, 451.
pp. 710-720.
ISSN 0304-8853
(2018)
Kırmızıbekmez Hasan; Kúsz Norbert; Bérdi Péter; Zupkó István; Hohmann Judit:
New iridoids from the roots of Valeriana dioscoridis Sm.
FITOTERAPIA, 130.
pp. 73-78.
ISSN 0367-326X
(2018)
Vágvölgyi Máté; Martins Ana; Kulmány Ágnes Erika; Zupkó István; Gáti Tamás; Simon András; Tóth Gábor; Hunyadi Attila:
Nitrogen-containing ecdysteroid derivatives vs. multi-drug resistance in cancer: preparation and antitumor activity of oximes, oxime ethers and a lactam.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 144.
pp. 730-739.
ISSN 0223-5234
(2018)
Bús Csaba; Kúsz Norbert; Jakab Gusztáv; Senobar Tahaei Seyyed Ashkan; Zupkó István; Endrész Valéria; Bogdanov Anita; Burián Katalin; Csupor-Löffler Boglárka; Hohmann Judit; Vasas Andrea:
Phenanthrenes from Juncus compressus Jacq. with promising antiproliferative and anti-HSV-2 activities.
MOLECULES, 23 (8).
Terjedelem: 13 p.-Azonosító: 2085.
ISSN 1420-3049
(2018)
Kiss Anita; Mernyák Erzsébet; Wölfling János; Sinka Izabella; Zupkó István; Schneider Gyula:
Stereoselective synthesis of the four 16-hydroxymethyl-3-methoxy- and 16-
hydroxymethyl-3-benzyloxy-13α-estra-1,3,5(10)-trien-17-ol isomers and
their antiproliferative activities.
STEROIDS, 134.
pp. 67-77.
ISSN 0039-128X
(2018)
Gonda Tímea; Bérdi Péter; Zupkó István; Fülöp Ferenc; Szakonyi Zsolt:
Stereoselective synthesis, synthetic and pharmacological application of monoterpene-based 1,2,4- and 1,3,4-oxadiazoles.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 19 (1).
Terjedelem: 11 p.-Azonosító: 81.
ISSN 1661-6596
(2018)
Minorics Renáta; Zupkó István:
Steroidal anticancer agents: an overview of estradiol-related compounds.
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, 18 (5).
pp. 652-666.
ISSN 1871-5206
(2018)
Le Tam Minh; Bérdi Péter; Zupkó István; Fülöp Ferenc; Szakonyi Zsolt:
Synthesis and transformation of (-)-isopulegol-based chiral β-aminolactones and β-aminoamides.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 19 (11).
Terjedelem: 19 p.-Azonosító: 3522.
ISSN 1661-6596
(2018)
Froehlich Tony; Kiss Anita; Wölfling János; Mernyák Erzsébet; Kulmány Ágnes Erika; Minorics Renáta; Zupkó István; Leidenberger Maria; Friedrich Oliver; Kappes Barbara; Hahn Friedrich; Marschall Manfred; Schneider Gyula; Tsogoeva Svetlana B.:
Synthesis of Artemisinin-Estrogen Hybrids Highly Active against HCMV, P-falciparum, and Cervical and Breast Cancer.
ACS MEDICINAL CHEMISTRY LETTERS, 9 (11).
pp. 1128-1133.
ISSN 1948-5875
(2018)
Pasinszki Tibor; Dzsotján Dániel; Lajgut Győző György; Harmat Veronika; Bor Andrea; Zupkó István; Csámpai Antal:
Synthesis, spectral- and theoretical study, x-ray analysis, and antiproliferative activity of 4,5-dihydrobenzoferroceno[1,2-d][1,2,3] selenadiazole and its benzo-fused analogue.
JOURNAL OF ORGANOMETALLIC CHEMISTRY, 863.
pp. 70-76.
ISSN 0022-328X
(2018)
Tóth Barbara; Kúsz Norbert; Forgó Péter; Bózsity Noémi; Zupkó István; Pinke Gyula; Hohmann Judit; Vasas Andrea:
Abietane diterpenoids from Sideritis montana L. and their antiproliferative activity.
FITOTERAPIA, 122.
pp. 90-94.
ISSN 0367-326X
(2017)
Roza Orsolya; Lai Wanchun; Zupkó István; Hohmann Judit; Jedlinszki Nikoletta; Chang Fang-Rong; Csupor Dezső; Eloff Jacobus Nicholaas:
Bioactivity guided isolation of phytoestrogenic compounds from Cyclopia genistoides by the pER8: GUS reporter system.
SOUTH AFRICAN JOURNAL OF BOTANY, 110.
pp. 201-207.
ISSN 0254-6299
(2017)
Kovács Bernadett; Béni Zoltán; Dékány Miklós; Orbán-Gyapai Orsolya; Sinka Izabella; Zupkó István; Hohmann Judit; Ványolós Attila:
Chemical analysis of the edible mushroom Tricholoma populinum: steroids and sulfinyladenosine compounds.
NATURAL PRODUCT COMMUNICATIONS, 12 (10).
pp. 1583-1584.
ISSN 1934-578X
(2017)
Baji Ádám; Kovács Ferenc; Mótyán Gergő; Schneider Gyula; Wölfling János; Sinka Izabella; Zupkó István; Ocsovszki Imre; Nagyné Frank Éva:
Investigation of pH and substituent effects on the distribution ratio of novel steroidal ring D- and A-fused arylpyrazole regioisomers and evaluation of their cell-growth inhibitory effects in vitro.
STEROIDS, 126.
pp. 35-49.
ISSN 0039-128X
(2017)
Laczkó-Zöld Eszter; Forgó Péter; Zupkó István; Sigrid Eşianu; Hohmann Judit:
Isolation and quantitative analysis of physalin D in the fruit and calyx of Physalis alkekengi L.
ACTA BIOLOGICA HUNGARICA, 68 (3).
pp. 300-309.
ISSN 0236-5383
(2017)
Bózsity Noémi; Minorics Renáta; Szabó Johanna; Mernyák Erzsébet; Schneider Gyula; Wölfling János; Wang Hui-Chun; Wu Chin-Chung; Ocsovszki Imre; Zupkó István:
Mechanism of antiproliferative action of a new D-secoestrone-triazole derivative in cervical cancer cells and its effect on cancer cell motility.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 165.
pp. 247-257.
ISSN 0960-0760
(2017)
Szakonyi Zsolt; Zupkó István; Fülöp Ferenc:
Stereoselective Synthesis and Antiproliferative Activity of Monoterpene-Fused 2-Imino-1,3-oxazines.
Current Organic Synthesis, 14 (4).
pp. 612-619.
ISSN 1570-1794
(2017)
Csomós Péter; Fodor Lajos; Zupkó István; Csámpai Antal; Sohár Pál:
Synthesis and in vitro antiproliferative effect of isomeric analogs of cyclobrassinin phytoalexin possessing the 1,3-thiazino[5,6-b]indole-4-one skeleton.
ARKIVOC, 4.
pp. 1-11.
ISSN 1551-7004
(2017)
Bodnár Brigitta; Mernyák Erzsébet; Szabó Johanna; Wölfling János; Schneider Gyula; Zupkó István; Kupihár Zoltán; Kovács Lajos:
Synthesis and in vitro investigation of potential antiproliferative monosaccharide-D-secoestrone bioconjugates.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 27 (9).
pp. 1938-1942.
ISSN 0960-894X
(2017)
Zupkó István:
A Szegedi Tudományegyetem Gyógyszerésztudományi Karán folyó tudományos munka bemutatása.
GYÓGYSZERÉSZET, 61 (11).
pp. 652-654.
ISSN 0017-6036
(2017)
Oprean Camelia; Zambori Csilla; Borcan Florin; Soica Codruta; Zupkó István; Minorics Renáta; Bojin Florina; Ambrus Rita; Muntean Delia; Danciu Corina; Pinzaru Iulia Andreea; Dehelean Cristina; Paunescu Virgil; Tanasie Gabriela:
Anti-proliferative and antibacterial in vitro evaluation of the polyurethane nanostructures incorporating pentacyclic triterpenes.
PHARMACEUTICAL BIOLOGY, 54 (11).
pp. 2714-2722.
ISSN 1388-0209
(2016)
Schelz Zsuzsanna; Ocsovszki Imre; Bózsity Noémi; Hohmann Judit; Zupkó István:
Antiproliferative Effects of Various Furanoacridones Isolated from Ruta graveolens on Human Breast Cancer Cell Lines.
ANTICANCER RESEARCH, 36 (6).
pp. 2751-2758.
ISSN 0250-7005
(2016)
Gospodinova Zlatina; Bózsity Noémi; Nikolova Milena T.; Krasteva Maria; Zupkó István:
Antiproliferative properties against human breast, cervical and ovarian cancer cell lines, and antioxidant capacity of leaf aqueous ethanolic extract from Cotinus coggygria Scop.
Acta Medica Bulgarica, 44 (2).
pp. 20-25.
ISSN 0324-1750
(2016)
Kuo Ching-Ying; Zupkó István; Chang Fang-Rong; Hunyadi Attila; Wu Chin-Chung; Weng Teng-Song; Wang Hui-Chun:
Dietary flavonoid derivatives enhance chemotherapeutic effect by inhibiting the DNA damage response pathway.
TOXICOLOGY AND APPLIED PHARMACOLOGY, 311.
pp. 99-105.
ISSN 0041-008X
(2016)
Antal Diana Simona; Ardelean Florina; Pinzaru Iulia; Borcan Florin; Ledeţi Ionuţ; Coricovac Dorina; Zupkó István; Baghdikian Beatrice; Ollivier Evelyne; Soica Codruta; Bolinitineanu Sorin Lucian:
Effects of cyclodextrin complexation on the anti-cancer effects of Cotinus coggygria extract and its constituents, butein and sulfuretin.
REVISTA DE CHIMIE, 67 (8).
pp. 1618-1622.
ISSN 0034-7752
(2016)
Andor Bogdan; Danciu Corina; Alexa Ersilia; Zupkó István; Hogea Elena; Cioca Andreea; Coricovac Dorina; Pinzaru Iulia; Pstrascu Jenel Marian; Mioc Marius; Cristina Romeo Teodor; Soica Codruta; Dehelean Cristina:
Germinated and Ungerminated Seeds Extract from Two Lupinus Species: Biological Compounds Characterization and In Vitro and In Vivo Evaluations.
EVIDENCE-BASED COMPLEMENTARY AND ALTERNATIVE MEDICINE, 2016.
Terjedelem: 8 p.-Azonosító: 7638542.
ISSN 1741-427X
(2016)
Ványolós Attila; Dékány Miklós; Kovács Bernadett; Krámos Balázs; Bérdi Péter; Zupkó István; Hohmann Judit; Béni Zoltán:
Gymnopeptides A and B, Cyclic Octadecapeptides from the Mushroom Gymnopus fusipes.
ORGANIC LETTERS, 18 (11).
pp. 2688-2691.
ISSN 1523-7060
(2016)
Molnár Judit; Szebeni Gábor J.; Csupor-Löffler Boglárka; Hajdú Zsuzsanna; Szekeres Thomas; Saiko Philipp; Ocsovszki Imre; Puskás László G.; Hohmann Judit; Zupkó István:
Investigation of the Antiproliferative Properties of Natural Sesquiterpenes from Artemisia asiatica and Onopordum acanthium on HL-60 Cells in Vitro.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 17 (2).
Terjedelem: 15 p.-Azonosító: 83.
ISSN 1661-6596
(2016)
Baji Ádám; Gyovai András; Wölfling János; Minorics Renáta; Ocsovszki Imre; Zupkó István; Nagyné Frank Éva:
Microwave-assisted one-pot synthesis of steroid–quinoline hybrids and an evaluation of their antiproliferative activities on gynecological cancer cell lines.
RSC ADVANCES, 6 (33).
pp. 27501-27516.
ISSN 2046-2069
(2016)
Mótyán Gergő; Kovács Ferenc; Wölfling János; Gyovai András; Zupkó István; Nagyné Frank Éva:
Microwave-assisted stereoselective approach to novel steroidal ring D-fused 2-pyrazolines and an evaluation of their cell-growth inhibitory effects in vitro.
STEROIDS, 112.
pp. 36-46.
ISSN 0039-128X
(2016)
Mótyán Gergő; Baji Ádám; Zupkó István; Nagyné Frank Éva:
Regio- and stereoselective synthesis of pregnane-fused isoxazolines by nitril-oxide/alkene 1,3-dipolar cycloaddition and an evaluation of their cell-growth inhibitory effect in vitro.
JOURNAL OF MOLECULAR STRUCTURE, 1110.
pp. 143-149.
ISSN 0022-2860
(2016)
Schneider Gyula; Kiss Anita; Mernyák Erzsébet; Benke Zsanett Amália; Wölfling János; Nagyné Frank Éva; Bózsity Noémi; Gyovai András; Minorics Renáta; Zupkó István:
Stereocontrolled synthesis of the four 16-hydroxymethyl-19-nortestosterone isomers and their antiproliferative activities.
STEROIDS, 105.
pp. 113-120.
ISSN 0039-128X
(2016)
Szabó Johanna; Pataki Zoltán; Wölfling János; Schneider Gyula; Bózsity Noémi; Minorics Renáta; Zupkó István; Mernyák Erzsébet:
Synthesis and biological evaluation of 13α-estrone derivatives as potential antiproliferative agents.
STEROIDS, 113.
pp. 14-21.
ISSN 0039-128X
(2016)
Bodnár Brigitta; Mernyák Erzsébet; Wölfling János; Schneider Gyula; Herman Bianka Edina; Szécsi Mihály; Sinka Izabella; Zupkó István; Kupihár Zoltán; Kovács Lajos:
Synthesis and biological evaluation of triazolyl 13α-estrone–nucleoside bioconjugates.
MOLECULES, 21 (9).
Paper 1212-16 p.
ISSN 1420-3049
(2016)
Szabó Johanna; Jerkovics Nóra; Schneider Gyula; Wölfling János; Bózsity Noémi; Minorics Renáta; Zupkó István; Mernyák Erzsébet:
Synthesis and in Vitro Antiproliferative Evaluation of C-13 Epimers of Triazolyl-d-Secoestrone Alcohols: The First Potent 13alpha-d-Secoestrone Derivative.
MOLECULES, 21 (5).
Terjedelem: 13 p.-Azonosító: 611.
ISSN 1420-3049
(2016)
Csábi József; Martins Ana; Sinka Izabella; Csorba Attila; Molnár József; Zupkó István; Tóth Gábor; Tillekeratne L. M. V.; Hunyadi Attila:
Synthesis and in vitro evaluation of the antitumor potential and chemo-sensitizing activity of fluorinated ecdysteroid derivatives.
MEDCHEMCOMM, 7 (12).
pp. 2282-2289.
ISSN 2040-2503
(2016)
Szabó Johanna; Bacsa Ildikó; Wölfling János; Schneider Gyula; Zupkó István; Varga Mónika; Herman Bianka Edina; Kalmár László; Szécsi Mihály; Mernyák Erzsébet:
Synthesis and in vitro pharmacological evaluation of N-[(1-benzyl-1,2,3-triazol-4-yl)methyl]-carboxamides on d-secoestrone scaffolds.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 31 (4).
pp. 574-579.
ISSN 1475-6366
(2016)
Kovács Dóra Irén; Wölfling János; Szabó Nikoletta; Szécsi Mihály; Schelz Zsuzsanna; Zupkó István; Nagyné Frank Éva:
Synthesis of novel 17-(4′-formyl)pyrazolylandrosta-5,16-dienes and their derivatives as potent 17α-hydroxylase/C17,20-lyase inhibitors or antiproliferative agents depending on the substitution pattern of the heteroring.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 120.
pp. 284-295.
ISSN 0223-5234
(2016)
Ványolós Attila; Kovács Bernadett; Bózsity Noémi; Zupkó István; Hohmann Judit:
Antiproliferative Activity of Some Higher Mushrooms from Hungary against Human Cancer Cell Lines.
INTERNATIONAL JOURNAL OF MEDICINAL MUSHROOMS, 17 (12).
pp. 1145-1149.
ISSN 1521-9437
(2015)
Gospodinova Zlatina; Bózsity Noémi; Ocsovszki Imre; Orbán-Gyapai Orsolya; Krasteva Maria; Zupkó István:
Chloroformic fraction of Tanacetum vulgare L. induces cell cycle arrest and apoptosis in MCF7 cells.
INTERNATIONAL JOURNAL OF PHARMA SCIENCES, 5 (2).
pp. 986-990.
ISSN 2320-6810
(2015)
Molnár Judit; Nagyné Frank Éva; Minorics Renáta; Kádár Zalán; Ocsovszki Imre; Schönecker Bruno; Wölfling János; Zupkó István:
A Click Approach to Novel D-Ring-Substituted 16α-Triazolylestrone Derivatives and Characterization of Their Antiproliferative Properties.
PLOS ONE, 10 (2).
Terjedelem: 27 p.-Azonosító: e0118104.
ISSN 1932-6203
(2015)
Kovács Dóra Irén; Wölfling János; Szabó Nikoletta; Szécsi Mihály; Minorics Renáta; Zupkó István; Nagyné Frank Éva:
Efficient access to novel androsteno-17-(1′,3′,4′)-oxadiazoles and 17<beta>-(1′,3′,4′)-thiadiazoles via N-substituted hydrazone and N,N′-disubstituted hydrazine intermediates, and their pharmacological evaluation in vitro.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 98.
pp. 13-22.
ISSN 0223-5234
(2015)
Rédei Dóra; Kúsz Norbert; Szabó Máté; Pinke Gyula; Zupkó István; Hohmann Judit:
First phytochemical investigation of secondary metabolites of Euphorbia davidii Subils. and antiproliferative activity of its extracts.
Acta Biologica Hungarica, 66 (4).
pp. 464-467.
ISSN 0236-5383
(2015)
Szekeres Márta; Nyergesné Illés Erzsébet; Janko Christina; Farkas Katalin; Tóth Ildikó; Nesztor Dániel; Zupkó István; Földesi Imre; Alexiou Christoph; Csákiné Tombácz Etelka:
Hemocompatibility and Biomedical Potential of Poly(gallic acid) Coated Iron Oxide Nanoparticles for Theranostic use.
JOURNAL OF NANOMEDICINE & NANOTECHNOLOGY, 6 (1).
Terjedelem: 7 p. -Azonosító: 1000252.
(2015)
Danciu Corina; Citu Cosmin; Zupkó István; Ghiulai Roxana; Matusz Petru; Pavel Zinuca Ioana; Popescu Alexandra; Pinzaru Iulia; Simu Georgeta; Daliborca Vlad C:
In vitro antiproliferative activity of flavonols: Fisetin, quercetin and kaempferol and their cyclodextrin complexes.
FARMACIA (BUCHAREST), 63 (6).
pp. 858-864.
ISSN 0014-8237
(2015)
Mótyán Gergő; Zupkó István; Minorics Renáta; Schneider Gyula; Wölfling János; Nagyné Frank Éva:
Lewis acid-induced intramolecular access to novel steroidal ring D-condensed arylpyrazolines exerting in vitro cell-growth-inhibitory effects.
MOLECULAR DIVERSITY, 19.
pp. 511-527.
ISSN 1381-1991
(2015)
Kiss Izabella; Vasas Andrea; Lajter Ildikó; Zupkó István; Hohmann Judit; Krupitza Georg:
Lobatin b inhibits NPM/ALK and NF-κB attenuating anaplastic-large-cell-lymphomagenesis and lymphendothelial tumour intravasation.
CANCER LETTERS, 356 (2 (Part B)).
pp. 994-1006.
ISSN 0304-3835
(2015)
Danciu Corina; Borcan Florin; Soica Codruta; Zupkó István; Csányi Erzsébet; Ambrus Rita; Muntean Delia; Sass Camelia; Antal Diana; Toma Claudia; Dehelean Cristina:
Polyurethane Microstructures-a Good or Bad in vitro Partner for the Isoflavone Genistein?
NATURAL PRODUCT COMMUNICATIONS, 10 (6).
pp. 951-954.
ISSN 1934-578X
(2015)
Danciu Corina; Soica Codruta; Dehelean Cristina; Zupkó István; Csányi Erzsébet; Pinzaru Iulia:
Preliminary In Vitro Evaluation of Genistein Chemopreventive Capacity as a Result of Esterification and Cyclodextrin Encapsulation.
ANALYTICAL CELLULAR PATHOLOGY, 2015.
Terjedelem: 8 p.-Azonosító: 262930.
ISSN 2210-7177
(2015)
Ledeţi Ionuţ; Avram Ştefana; Bercean Vasile; Vlase Gabriela; Vlase Titus; Ledeti Adriana; Zupkó István; Mioc Marius; Suta Lenuta-Maria; Soica Codruta; Dehelean Cristina:
Solid-State Characterization and Biological Activity of Betulonic Acid Derivatives.
MOLECULES, 20 (12).
pp. 22691-22702.
ISSN 1420-3049
(2015)
Palici Ionut F.; Liktor-Busa Erika; Zupkó István; Touzard Blaise; Chaieb Mohamed; Zsoldiné Urbán Edit; Hohmann Judit:
Study of in vitro antimicrobial and antiproliferative activities of selected Saharan plants.
ACTA BIOLOGICA HUNGARICA, 66 (4).
pp. 385-394.
ISSN 0236-5383
(2015)
Huber Imre; Zupkó István; Kovács Ida Jusztina; Minorics Renáta; Gulyás Gergely; Maász Gábor; Perjési Pál:
Synthesis and Antiproliferative Activity of Cyclic Arylidene Ketones: Direct Comparison of Monobenzylidene and Dibenzylidene Derivatives.
MONATSHEFTE FUR CHEMIE, 146 (6).
pp. 973-981.
ISSN 0026-9247
(2015)
Huber Judit; Wölfling János; Schneider Gyula; Ocsovszki Imre; Varga Mónika; Zupkó István; Mernyák Erzsébet:
Synthesis of antiproliferative 13α-d-homoestrones via Lewis acid-promoted one-pot Prins–Ritter reactions of d-secosteroidal δ-alkenyl-aldehydes.
STEROIDS, 102.
pp. 76-84.
ISSN 0039-128X
(2015)
Szabó Nikoletta; Iványi Zoltán; Szécsi Mihály; Julesz János; Mernyák Erzsébet; Huber Judit; Wölfling János; Minorics Renáta; Zupkó István; Schneider Gyula:
Synthesis of methoxycarbonylpyrazolylandrostene derivatives, and their potential inhibitory effect on androgen biosynthesis and cell proliferation.
Steroids, 98.
pp. 143-152.
ISSN 0039-128X
(2015)
Schneider Gyula; Görbe Tamás Ferenc; Mernyák Erzsébet; Wölfling János; Holczbauer Tamás; Czugler Mátyás; Sohár Pál; Minorics Renáta; Zupkó István:
Synthesis of novel 17-(5’-iodo)triazolyl-3-methoxyestrane epimers via Cu(I)-catalyzed azide-alkyne cycloadditon, and an evaluation of their cytotoxic activity in vitro.
STEROIDS, 98.
pp. 153-165.
ISSN 0039-128X
(2015)
Mernyák Erzsébet; Kovács Ida; Minorics Renáta; Sere Péter; Czégány Dóra; Sinka Izabella; Wölfling János; Schneider Gyula; Újfaludi Zsuzsanna; Boros Imre Miklós; Ocsovszki Imre; Varga Mónika; Zupkó István:
Synthesis of trans-16-triazolyl-13α-methyl-17-estradiol diastereomers and the effects of structural modifications on their in vitro antiproliferative activities.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 150.
pp. 123-134.
ISSN 0960-0760
(2015)
Blaschke Michael; McKinnon Ruxandra; Huu Chi Nguyen; Holzner Silvio; Zehl Martin; Atanasov Atanas Georgiev; Schelch Karin; Krieger Sigurd; Diaz Rene; Frisch Richard; Feistel Björn; Jäger Walter; Ecker Gerhard F; Dirsch Verena M; Grusch Michael; Zupkó István; Urban Ernst; Kopp Brigitte; Krupitza Georg:
A eudesmane-type sesquiterpene isolated from Pluchea odorata (L.) Cass. combats three hallmarks of cancer cells: unrestricted proliferation, escape from apoptosis and early metastatic outgrowth in vitro.
MUTATION RESEARCH-FUNDAMENTAL AND MOLECULAR MECHANISMS OF MUTAGENESIS, 777.
pp. 79-90.
ISSN 0027-5107
(2015)
Unger Christine; Kiss Izabella; Vasas Andrea; Lajter Ildikó; Zupkó István; Hohmann Judit; Krupitza Georg:
The germacranolide sesquiterpene lactone neurolenin B of the medicinal plant Neurolaena lobata (L.) R.Br. ex Cass inhibits NPM/ALK-driven cell expansion and NF-κB-driven tumour intravasation.
PHYTOMEDICINE, 22 (9).
pp. 862-874.
ISSN 0944-7113
(2015)
İstanbullu Huseyin; Zencir Sevil; Berényi Ágnes; Canturk Kilikaya Pakize; Zupkó István; Erciyas Ercin; Topcu Zeki:
The interference of piperidinopropionaphthone hydrochloride in mammalian type I and type II DNA topoisomerase reactions.
MARMARA ECZACILIK DERGISI / MARMARA PHARMACEUTICAL JOURNAL, 19 (2).
pp. 82-87.
ISSN eISSN: 1309-0801
(2015)
Minorics Renáta; Bózsity Noémi; Molnár Judit; Wölfling János; Mernyák Erzsébet; Schneider Gyula; Ocsovszki Imre; Zupkó István:
A molecular understanding of d-homoestrone-induced G2/M cell cycle arrest in HeLa human cervical carcinoma cells.
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 19 (10).
pp. 2365-2374.
ISSN 1582-1838
(2015)
Kúsz Norbert; Rédei Dóra; Blazsó Gábor; Jedlinszki Nikoletta; Zupkó István; Hohmann Judit:
Anti-inflammatory effect of sea-buckthorn fruit in vivo.
Planta Medica, 80 (16).
P1L6-P1L6.
ISSN 0032-0943
(2014)
Zupkó István; Molnár Judit; Réthy Borbála; Minorics Renáta; Nagyné Frank Éva; Wölfling János; Molnár József; Ocsovszki Imre; Topcu Zeki; Bitó Tamás; Puskás László:
Anticancer and multidrug resistance-reversal effects of solanidine analogs synthetized from pregnadienolone acetate.
MOLECULES, 19 (2).
pp. 2061-2076.
ISSN 1420-3049
(2014)
Hajdú Zsuzsanna; Hohmann Judit; Forgó Péter; Máthé Imre; Molnár Judit; Zupkó István:
Antiproliferative Activity of Artemisia asiatica Extract and Its Constituents on Human Tumor Cell Lines.
Planta Medica, 80 (18).
pp. 1692-1697.
ISSN 0032-0943
(2014)
Hajdú Zsuzsanna; Hohmann Judit; Forgó Péter; Máthé Imre; Molnár Judit; Zupkó István:
Antiproliferative activity of Artemisia asiatica cultivated in Central Europe.
Planta Medica, 80 (16).
P2B30-P2B30.
ISSN 0032-0943
(2014)
Soica Codruta; Danciu Corina; Savoiu-Balint Germaine; Borcan Florin; Ambrus Rita; Zupkó István; Bojin Florina; Coricovac Dorina; Ciurlea Sorina; Avram Ştefana; Dehelean Cristina Adriana; Olariu Teodora; Matusz Petru:
Betulinic Acid in Complex with a Gamma-Cyclodextrin Derivative Decreases Proliferation and in Vivo Tumor Development of Non-Metastatic and Metastatic B164A5 Cells.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 15 (5).
pp. 8235-8255.
ISSN 1661-6596
(2014)
Csupor-Löffler Boglárka; Zupkó István; Molnár Judit; Forgó Péter; Hohmann Judit:
Bioactivity-guided isolation of antiproliferative compounds from the roots of Onopordum acanthium.
Natural Product Communications, 9 (3).
pp. 337-340.
ISSN 1934-578X
(2014)
Trandafirescu Cristina; Antal Diana; Soica Codruta; Zupkó István; Minorics Renáta; Ambrus Rita; Borcan Florin; Oprean Camelia; Danciu Corina; Avram Ştefana; Dehelean Cristina; Nita Simona; Vlaia Lavinia:
Cyclodextrin Complexes of Oleanolic and Ursolic Acid: Physico-chemical and biological preliminary evaluation.
REVISTA DE CHIMIE, 65 (10).
pp. 1163-1167.
ISSN 0034-7752
(2014)
Danciu Corina; Soica Codruta; Oltean Mircea; Avram Ştefana; Borcan Florin; Csányi Erzsébet; Ambrus Rita; Zupkó István; Muntean Muntean; Dehelean Cristina A.; Craina Marius; Popovici Ramona A.:
Genistein in 1:1 inclusion complexes with ramified cyclodextrins: theoretical, physicochemical and biological evaluation.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 15 (2).
pp. 1962-1982.
ISSN 1661-6596
(2014)
Kúsz Norbert; Rédei Dóra; Blazsó Gábor; Jedlinszki Nikoletta; Hohmann Judit; Zupkó István:
Homoktövitermés-kivonat gyulladásgátló hatásának értékelése in vivo.
Gyógyszerészet, 58 (Suppl 1).
p. 86.
ISSN 0017-6036
(2014)
Ványolós Attila; Zupkó István; Kovács Bernadett; Hohmann Judit:
Investigation of the antiproliferative activity of some higher macrofungi.
CHEMICKE LISTY, 108.
s144-s145.
ISSN 0009-2770
(2014)
Sztojkov-Ivanov Anita; Szolomájer-Csikos Orsolya; Márki Árpád; Tóth Gábor; Zupkó István:
Investigation of the pharmacokinetics of the ABCG2 transporter inhibitor Ko134 in mice by a newly developed and validated HPLC method.
CURRENT PHARMACEUTICAL ANALYSIS, 10 (1).
pp. 30-37.
ISSN 1573-4129
(2014)
Lajter Ildikó; Vasas Andrea; Béni Zoltán; Forgó Péter; Binder Markus; Bochkov Valery; Zupkó István; Krupitza Georg; Frisch Richard; Kopp Brigitte; Hohmann Judit:
Isolation and characterisation of new bioactive compounds from Neurolaena lobata.
CHEMICKE LISTY, 108.
s135-s135.
ISSN 0009-2770
(2014)
Berkó Szilvia; Balázs Boglárka; Sütő Blanka; Erős Gábor; Gál Brigitta; Sztojkov-Ivanov Anita; Codruta Soica; Révész Piroska; Kemény Lajos; Zupkó István; Csányi Erzsébet:
Monitoring of skin penetration and absorption with a new in vivo experimental model.
FARMACIA, 62 (6).
pp. 1157-1163.
ISSN 0014-8237
(2014)
Molnár Judit; Hajdú Zsuzsanna; Csupor-Löffler Boglárka; Szekeres Thomas; Saiko Philipp; Ocsovszki Imre; Hohmann Judit; Zupkó István:
Növényi eredetű szeszkviterpének tumorellenes hatásának vizsgálata in vitro.
Gyógyszerészet, 58 (Suppl 1).
p. 98.
ISSN 0017-6036
(2014)
McKinnon Ruxandra; Binder Markus; Zupkó István; Afonyushkin Taras; Lajter Ildikó; Vasas Andrea; de Martin Rainer; Unger Christine; Dolznig Helmut; Diaz Rene; Risch Richard; Passreiter Claus M.; Krupitza Georg; Hohmann Judit; Kopp Brigitte; Bochkov Valery N.:
Pharmacological insight into the anti-inflammatory activity of sesquiterpene lactones from Neurolaena lobata (L.) R.Br. ex Cass.
PHYTOMEDICINE, 21 (12).
pp. 1695-1701.
ISSN 0944-7113
(2014)
Jedlinszki Nikoletta; Rédei Dóra; Haller József; Freund Tamás F; Hohmann Judit; Zupkó István:
Possible role of fat tissue in the pharmacokinetics of dodeca-2E,4E,8Z,10E/ Z-tetraenoic acid isobutylamides after oral administration of Echinacea angustifolia extract in rats.
Natural Product Communications, 9 (6).
pp. 843-845.
ISSN 1934-578X
(2014)
Lajter Ildikó; Vasas Andrea; Béni Zoltán; Forgó Péter; Binder Markus; Bochkov Valery; Zupkó István; Krupitza Georg; Frisch Richard; Kopp Brigitte; Hohmann Judit:
Sesquiterpenes from Neurolaena lobata and Their Antiproliferative and Anti-inflammatory Activities.
Journal of Natural Products, 77 (3).
pp. 576-582.
ISSN 0163-3864
(2014)
Szakonyi Zsolt; Zupkó István; Sillanpää Reijo; Fülöp Ferenc:
Stereoselective Synthesis and Cytoselective Toxicity of Monoterpene-Fused 2-Imino-1,3-thiazines.
Molecules, 19 (10).
pp. 15918-15937.
ISSN 1420-3049
(2014)
Mernyák Erzsébet; Szabó Johanna; Bacsa Ildikó; Huber Judit; Schneider Gyula; Minorics Renáta; Bózsity Noémi; Zupkó István; Varga Mónika; Bikádi Zsolt; Hazai Eszter; Wölfling János:
Syntheses and Antiproliferative Effects of D-homo- and D-secoestrones.
STEROIDS, 87.
pp. 128-136.
ISSN 0039-128X
(2014)
Mernyák Erzsébet; Fiser Gabriella; Szabó Johanna; Bodnár Brigitta; Schneider Gyula; Kovács Ida Jusztina; Ocsovszki Imre; Zupkó István; Wölfling János:
Synthesis and in vitro antiproliferative evaluation of D-secooxime derivatives of 13β- and 13α-estrone.
STEROIDS, 89.
pp. 47-55.
ISSN 0039-128X
(2014)
Nagyné Frank Éva; Kovács Dóra Irén; Schneider Gyula; Wölfling János; Bartók Tibor; Zupkó István:
Synthesis of novel steroidal 16-spiroisoxazolines by 1,3-dipolar cycloaddition, and an evaluation of their antiproliferative activities in vitro.
MOLECULAR DIVERSITY, 18 (3).
pp. 521-534.
ISSN 1381-1991
(2014)
Kovács Dóra; Mótyán Gergő; Wölfling János; Kovács Ida; Zupkó István; Frank Éva:
A facile access to novel steroidal 17-2′-(1′,3′,4′)-oxadiazoles, and an evaluation of their cytotoxic activities in vitro.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 24.
pp. 1265-1268.
ISSN 0960-894X
(2014)
Lajter Ildikó; Zupkó István; Molnár Judit; Jakab Gusztáv; Balogh Lajos; Vasas Andrea; Hohmann Judit:
Antiproliferative Activity of Polygonaceae Species from the Carpathian Basin against Human Cancer Cell Lines.
Phytotherapy Research, 27 (1).
pp. 77-85.
ISSN 0951-418X
(2013)
Hohmann Judit; Rédei Dóra; Kúsz Norbert; Jedlinszki Nikoletta; Forgó Péter; Blazsó Gábor; Zupkó István:
Bioactivity-guided isolation of anti-inflammatory constituents from the fruits of buckthorn (Hippophae rhamnoides).
In:
VI. International Conference on Polyphenols and Health. Buenos Aires, Argentína, 2013.10.16-2013.10.19.
ICPH, p. 49.
(2013)
Bourgonje Vincent J.A.; Vos Marc A.; Ozdemir Semir; Doisne Nicolas; Acsai Károly; Varró András; Sztojkov-Ivanov Anita; Zupkó István; Rauch Erik; Kattner Lars; Bito Virginie; Houtman Marien; Nagel, van der Roel; Beekman Jet D.; Veen, van Toon A.B.; Sipido Karin R.; Antoons Gudrun:
Combined Na+/Ca2+ Exchanger and L-Type Calcium Channel Block as a Potential Strategy to Suppress Arrhythmias and Maintain Ventricular Function.
CIRCULATION-ARRHYTHMIA AND ELECTROPHYSIOLOGY, 6 (2).
pp. 371-379.
ISSN 1941-3149
(2013)
Mernyák Erzsébet; Huber Judit; Szabó Johanna; Schneider Gyula; Hetényi Anasztázia; Márk László; Maász Gábor; Berényi Ágnes; Kovács Ida Jusztina; Minorics Renáta; Zupkó István; Wölfling János:
Cycloaddition of Steroidal Cyclic Nitrones to C=N Dipolarophiles: Stereoselective Synthesis and Antiproliferative Effects of Oxadiazolidinones in the Estrone Series.
STEROIDS, 78 (10).
pp. 1021-1028.
ISSN 0039-128X
(2013)
Hunyadi Attila; Veres Katalin; Dankó Balázs Ödön; Kele Zoltán; Wéber Edit; Hetényi Anasztázia; Zupkó István; Hsieh Tusty-Jiuan:
In vitro Anti-diabetic Activity and Chemical Characterization of an Apolar Fraction of Morus alba Leaf Water Extract.
Phytotherapy Research, 27 (6).
pp. 847-851.
ISSN 0951-418X
(2013)
Molnár Judit; Ocsovszki Imre; Puskás László; Ghane Tannaz; Hohmann Judit; Zupkó István:
Investigation of the antiproliferative action of the quinoline alkaloids kokusaginine and skimmianine on human cell lines.
Current Signal Transduction Therapy, 8 (2).
pp. 148-155.
ISSN 1574-3624
(2013)
Hunyadi Attila; Liktor-Busa Erika; Márki Árpád; Martins Ana; Jedlinszki Nikoletta; Hsieh T. J.; Báthori Mária; Hohmann Judit; Zupkó István:
Metabolic effects of mulberry leaves: Exploring potential benefits in type 2 diabetes and hyperuricemia.
Evidence-Based Complementary and Alternative Medicine.
Azonosító: N°948627-Terjedelem: 11 p..
ISSN 1741-427X
(2013)
Jedlinszki Nikoletta; Rédei Dóra; Haller József; Freund Tamás F; Hohmann Judit; Zupkó István:
Pharmacokinetics of dodeca-2E,4E,8Z,10E/Z-tetraenoic acid isobutylamides after oral administration of Echinacea angustifolia extract in rats.
In:
9th Balaton Symposium on High-Performance Separation Methods. Siófok, Magyarország, 2013.09.04-2013.09.06.
Hungarian Society for Separation Sciences, Pécs, p. 116.
(2013)
ISBN 978-963-89335-2-2
Roza Orsolya; Lovász Norbert; Zupkó István; Hohmann Judit; Csupor Dezső:
Sympathomimetic activity of a Hoodia gordonii product: a possible mechanism of cardiovascular side effects.
BioMed Research International.
Azonosító: N°171059-Terjedelem: 7 p..
ISSN 2314-6133
(2013)
Minorics Renáta; Bózsity Noémi; Wölfling János; Mernyák Erzsébet; Schneider Gyula; Márki Árpád; Falkay György; Ocsovszki Imre; Zupkó István:
Antiproliferative effect of normal and 13-epi-d-homoestrone and their 3-methyl ethers on human reproductive cancer cell lines.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 132.
pp. 168-175.
ISSN 0960-0760
(2012)
Forgó Péter; Zupkó István; Molnár Judit; Vasas Andrea; Dombi György; Hohmann Judit:
Bioactivity-guided isolation of antiproliferative compounds from Centaurea jacea L.
Fitoterapia, 83 (5).
pp. 921-925.
ISSN 0367-326X
(2012)
Hunyadi Attila; Martins Ana; Hsieh Tusty-Jiuan; Seres Adrienn; Zupkó István:
Chlorogenic acid and rutin play a major role in the in vivo anti-diabetic activity of Morus alba leaf extract on type II diabetic rats.
PLoS ONE, 7 (11).
Terjedelem: 6 p.-Azonosító: e50619.
ISSN 1932-6203
(2012)
Vasas Andrea; Sulyok Edvárd István; Martins Ana; Rédei Dóra; Forgó Péter; Kele Zoltán; Zupkó István; Molnár József; Pinke Gyula; Hohmann Judit:
Cyclomyrsinane and premyrsinane diterpenes from Euphorbia falcata modulate
resistance of cancer cells to doxorubicin.
Tetrahedron, 68 (4).
pp. 1280-1285.
ISSN 0040-4020
(2012)
Martins Ana; Tóth Noémi; Ványolós Attila; Béni Zoltán; Zupkó István; Molnár József; Báthori Mária; Hunyadi Attila:
Significant activity of ecdysteroids on the resistance to doxorubicin in mammalian cancer cells expressing the human ABCB1 transporter.
Journal of Medicinal Chemistry, 55 (11).
pp. 5034-5043.
ISSN 0022-2623
(2012)
Ndonsta Blanche L.; Tatsimo N. Simplice Joel; Csupor Dezső; Forgó Péter; Berkecz Róbert; Berényi Ágnes; Tene Mathieu; Molnár Judit; Zupkó István; Hohmann Judit; Tane Pierre:
Alkylbenzoquinones with antiproliferative effect against human cancer cell lines from stem of Ardisia kivuensis.
Phytochemistry Letters, 4 (3).
pp. 227-230.
ISSN 1874-3900
(2011)
Csupor-Löffler Boglárka; Hajdú Zsuzsanna; Zupkó István; Molnár Judit; Forgó Péter; Vasas Andrea; Kele Zoltán; Hohmann Judit:
Antiproliferative constituents of the roots of Conyza canadensis.
Planta Medica, 77 (11).
pp. 1183-1188.
ISSN 0032-0943
(2011)
Janicsák Gábor; Zupkó István; Nikolova Milena T.; Forgó Péter; Vasas Andrea; Máthé Imre; Blunden Gerald; Hohmann Judit:
Bioactivity-guided study of antiproliferative activities of Salvia extracts.
Natural Product Communications, 6 (5).
pp. 575-579.
ISSN 1934-578X
(2011)
Csupor Dezső; Borcsa Botond Lajos; Heydel Barbara; Hohmann Judit; Zupkó István; Ma Yan; Widowitz Ute; Bauer Rudolf:
Comparison of a specific HPLC determination of toxic aconite
alkaloids in processed Radix aconiti with a titration method of total alkaloids.
Pharmaceutical Biology, 49 (10).
pp. 1097-1101.
ISSN 1388-0209
(2011)
Vasas Andrea; Sulyok Edvárd István; Rédei Dóra; Forgó Péter; Szabó Pál Tamás; Zupkó István; Berényi Ágnes; Molnár József; Hohmann Judit:
Jatrophane diterpenes from Euphorbia esula as antiproliferative agents and potent chemosensitizers to overcome multidrug resistance.
Journal of Natural Products, 74 (6).
pp. 1453-1461.
ISSN 0163-3864
(2011)
Nagyné Frank Éva; Molnár Judit; Zupkó István; Kádár Zalán; Wölfling János:
Synthesis of novel steroidal 17α-triazolyl derivatives via Cu(I)-catalyzed azide-alkyne cycloaddition, and an evaluation of their cytotoxic activity in vitro.
STEROIDS, 76 (10-11).
pp. 1141-1148.
ISSN 0039-128X
(2011)
Fodor Lajos; Csomós Péter; Molnár Judit; Zupkó István; Csámpai Antal; Sohár Pál:
Unexpected formation of indenoisoquinoline derivatives from thia analogues of protoberberine alkaloids.
Letters in Organic Chemistry, 8 (7).
pp. 450-453.
ISSN 1570-1786
(2011)
Csapi Bence; Hajdú Zsuzsanna; Zupkó István; Berényi Ágnes; Forgó Péter; Szabó Pál Tamás; Hohmann Judit:
Bioactivity-guided isolation of antiproliferative compounds from Centaurea arenaria.
PHYTOTHERAPY RESEARCH, 24 (11).
pp. 1664-1669.
ISSN 0951-418X
(2010)
Hajdú Zsuzsanna; Zupkó István; Réthy Borbála; Forgó Péter; Hohmann Judit:
Bioactivity-guided isolation of cytotoxic sesquiterpenes and flavonoids from Anthemis ruthenica.
PLANTA MEDICA: NATURAL PRODUCTS AND MEDICINAL PLANT RESEARCH, 76 (1).
pp. 94-96.
ISSN 0032-0943
(2010)
Janicsák Gábor; Zupkó István; Máthé Imre; Hohmann Judit:
Comparative study of the antioxidant activities of eleven Salvia species.
NATURAL PRODUCT COMMUNICATIONS, 5 (2).
pp. 227-230.
ISSN 1934-578X
(2010)
Zupkó István:
A Hypericum perforatum kivonat antidepresszáns hatásának feltételezett mechanizmusa.
PHARMA ÉS FLÓRA - FITOTERÁPIÁS TOVÁBBKÉPZŐ FOLYÓIRAT, 1 (4).
pp. 8-10.
ISSN 2062-6231
(2010)
Nagyné Frank Éva; Mucsi Zoltán; Szécsi Mihály; Zupkó István; Wölfling János; Schneider Gyula:
Intramolecular approach to some new D-ring-fused steroidal isoxazolidines by 1,3-dipolar cycloaddition: synthesis, theoretical and in vitro pharmacological studies.
NEW JOURNAL OF CHEMISTRY, 34 (11).
pp. 2671-2681.
ISSN 1144-0546
(2010)
Csupor Dezső; Wenzig Eva Maira; Zupkó István; Wolkart Karin; Hohmann Judit; Bauer Rudolf:
Qualitative and quantitative analysis of aconitine-type and lipo-alkaloids of Aconitum carmichaelii roots.
JOURNAL OF CHROMATOGRAPHY A, 1216 (11).
pp. 2079-2086.
ISSN 0021-9673
(2009)
Kovács Adriána; Vasas Andrea; Forgó Péter; Réthy Borbála; Zupkó István; Hohmann Judit:
Xanthanolides with antitumour activity from Xanthium italicum.
ZEITSCHRIFT FÜR NATURFORSCHUNG C-A JOURNAL OF BIOSCIENCES, 64 (5-6).
pp. 343-349.
ISSN 0939-5075
(2009)
Háznagyné Radnai Erzsébet; Réthy Borbála; Czigle Szilvia; Zupkó István; Wéber Edit; Martinek Tamás A.; Falkay György; Máthé Imre:
Cytotoxic activities of Stachys species.
FITOTERAPIA, 79 (7-8).
pp. 595-597.
ISSN 0367-326X
(2008)
Csupor Dezső; Forgó Péter; Zupkó István; Szabó Pál Tamás; Hohmann Judit:
Anthranoyl-substituted norditerpene alkaloids from Aconitum vulpalia Rchb. and their cytotoxic activities.
ZEITSCHRIFT FUR NATURFORSCHUNG SECTION B-A JOURNAL OF CHEMICAL SCIENCES, 62 (1).
pp. 135-141.
ISSN 0932-0776
(2007)
Hajdú Zsuzsanna; Hohmann Judit; Forgó Péter; Martinek Tamás; Dervarics Mate; Zupkó István; Falkay György; Cossuta Dániel; Máthé Imre:
Diterpenoids and flavonoids from the fruits of Vitex agnus-castus and antioxidant activity of the fruit extracts and their constituents.
PHYTOTHERAPY RESEARCH, 21 (4).
pp. 391-394.
ISSN 0951-418X
(2007)
Báthori Mária; Zupkó István; Hunyadi Attila; Gacsne-Baitz Eszter; Dinya Zoltán; Forgó Péter:
Monitoring the antioxidant activity of extracts originated from various Serratula species and isolation of flavonoids from Serratula coronata.
FITOTERAPIA, 75 (2).
pp. 162-167.
ISSN 0367-326X
(2004)
Havass Judit; Bakos Krisztina; Márki Árpád; Gáspár Róbert; Gera Lajos; Fülöp Ferenc; Tóth Gábor; Zupkó István; Falkay György:
Noncompetitive nature of oxytocin antagonists with general structure Mpa(1)XXX(2)Sar(7)Arg(8).
PEPTIDES, 23 (8).
pp. 1419-1425.
ISSN 0196-9781
(2002)
Zupkó István; Márki Árpád; Gáspár Róbert; Falkay György:
Correlation between alpha 1/beta-adrenoceptor ratio and spontaneous uterine motor activity in the post-partum rat.
MOLECULAR HUMAN REPRODUCTION, 4 (9).
pp. 921-924.
ISSN 1360-9947
(1998)
Gáspár Róbert; Márki Árpád; Zupkó István; Falkay György:
Evidence of non-synaptic regulation of postpartum uterine contractility in the rat.
LIFE SCIENCES, 62 (12).
pp. 1119-1124.
ISSN 0024-3205
(1998)
Zupkó István; Gáspár Róbert; Kovács L.; Falkay György:
Are alpha-adrenergic antagonists potent tocolytics? In vivo experiments on postpartum rats.
LIFE SCIENCES, 61 (11).
PL159-PL163.
ISSN 0024-3205
(1997)
Zupkó István; Blazsó Gábor; Minker Emil:
Kalcium-csatorna blokkolók hatása patkány nervus phrenicus-diaphragma preparátum elektromos és mechanikus válaszára [Effects of calcium channel blockers on electrical and mechanical responses of rat phrenic nerve-diaphragm preparations].
ACTA PHARMACEUTICA HUNGARICA, 65 (4).
pp. 127-131.
ISSN 0001-6659
(1995)