Tayeb Bizhar Ahmed; Njangiru Isaac Kinyua; Minorics Renáta:
Beyond boundaries: Neuroprotective effects of steroids and ecdysteroids in SH‐SY5Y cells ‐ A systematic review.
NEUROPROTECTION, 2 (2).
pp. 151-166.
ISSN 2770-7296
(2024)
Gáborová Mária; Vágvölgyi Máté; Tayeb Bizhar Ahmed; Minorics Renáta; Zupkó István; Jurček Ondřej; Béni Szabolcs; Kubínová Renata; Balogh György Tibor; Hunyadi Attila:
Diterpenes Isolated from Three Different Plectranthus Sensu Lato Species and Their Antiproliferative Activities against Gynecological and Glioblastoma Cancer Cells.
ACS OMEGA, 9 (16).
pp. 18495-18504.
ISSN 2470-1343
(2024)
Tayeb Bizhar Ahmed; Kusuma Ikhwan Yuda; Osman Alaa Awadallah Mohammedalhassan; Minorics Renáta:
Herbal compounds as promising therapeutic agents in precision medicine strategies for cancer: A systematic review.
JOURNAL OF INTEGRATIVE MEDICINE, 22 (2).
pp. 137-162.
ISSN 2095-4964
(2024)
Szilvásy Nóra; Lajer Panna; Horváth Attila; Veres Katalin; Hohmann Judit; Schelz Zsuzsanna; Minorics Renáta; Zupkó István; Gáborik Zsuzsanna; Kis Emese; Temesszentandrási-Ambrus Csilla:
Modulation of Multispecific Transporters by Uncaria tomentosa Extract and Its Major Phytoconstituents.
PHARMACEUTICS, 16 (11).
ISSN 1999-4923
(2024)
Bózsity-Faragó Noémi; Nagy Viktória; Szabó Johanna; Pálházi Balázs; Kele Zoltán; Resch Vivien; Paragi Gábor; Zupkó István; Minorics Renáta; Mernyák Erzsébet:
Synthesis of Estrone Heterodimers and Evaluation of Their In Vitro Antiproliferative Activity.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 25 (8).
ISSN 1661-6596
(2024)
Ahmed Sara Hassan Hassan; Tayeb Bizhar Ahmed; Gonda Tímea; Girst Gábor; Szőri Kornél; Berkecz Róbert; Zupkó István; Minorics Renáta; Hunyadi Attila:
Thymoquinone-protoflavone hybrid molecules as potential antitumor agents.
PLOS ONE, 19 (1).
ISSN 1932-6203
(2024)
Senobar Tahaei Seyyed Ashkan; Kulmány Ágnes; Minorics Renáta; Kiss Anita; Szabó Zoltán; Germán Péter; Szebeni Gábor; Gémes Nikolett; Mernyák Erzsébet; Zupkó István:
Antiproliferative and Antimetastatic Properties of 16-Azidomethyl Substituted 3-O-Benzyl Estrone Analogs.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 24 (18).
ISSN 1661-6596
(2023)
Nagy Viktória; Mounir Raji; Szebeni Gábor J.; Szakonyi Zsolt; Gémes Nikolett; Minorics Renáta; Germán Péter; Zupkó István:
Investigation of Anticancer Properties of Monoterpene-Aminopyrimidine Hybrids on A2780 Ovarian Cancer Cells.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 24 (13).
ISSN 1661-6596
(2023)
Lőrincz Eszter Boglárka; Tóth Gergely; Spolárics Júlia; Herczeg Mihály; Hodek Jan; Zupkó István; Minorics Renáta; Ádám Dorottya; Oláh Attila; Zouboulis Christos C.; Weber Jan; Nagy Lajos; Ostorházi Eszter; Bácskay Ildikó; Borbás Anikó; Herczegh Pál; Bakai-Bereczki Ilona:
Mannich-type modifications of (−)-cannabidiol and (−)-cannabigerol leading to new, bioactive derivatives.
SCIENTIFIC REPORTS, 13 (1).
ISSN 2045-2322
(2023)
Kovács Édua; Ali Hazhmat; Minorics Renáta; Traj Péter; Resch Vivien Erzsébet; Paragi Gábor; Bruszel Bella; Zupkó István; Mernyák Erzsébet:
Synthesis and Antiproliferative Activity of Steroidal Diaryl Ethers.
MOLECULES, 28 (3).
ISSN 1420-3049
(2023)
Bamou Zahra Fatima; Le Minh Tam; Tayeb Bizhar Ahmed; Tahaei Seyyed Ashkan Senobar; Minorics Renáta; Zupkó István; Szakonyi Zsolt:
Antiproliferative Activity of (-)-Isopulegol-based 1,3-Oxazine, 1,3-Thiazine and 2,4-Diaminopyrimidine Derivative.
CHEMISTRYOPEN, 11 (10).
ISSN 2191-1363
(2022)
Molnár Barnabás; Njangiru Isaac Kinyua; Mótyán Gergő; Leits Péter; Zupkó István; Minorics Renáta; Balogh György Tibor; Nagyné Frank Éva:
Regioselective synthesis, physicochemical properties and anticancer activity of 2-aminomethylated estrone derivatives.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 219.
Terjedelem: 13 p-Azonosító: 106064.
ISSN 0960-0760
(2022)
Ristovski Jovana; Minorics Renáta; Bartha Sándor; Jankovic Nenad; Zupkó István:
The evaluation of the anticancer activity of the Biginelli hybrids and pharmacokinetic profiling based on their retention parameters.
Journal of Molecular Structure, 1254.
Terjedelem: 12-Azonosító: 132373.
ISSN 0022-2860
(2022)
Mernyák Erzsébet; Bartha Sándor; Kóczán Lili; Jójárt Rebeka; Resch Vivien; Paragi Gábor; Vágvölgyi Máté; Hunyadi Attila; Bruszel Bella; Zupkó István; Minorics Renáta:
Microwave-assisted Phospha-Michael addition reactions in the 13 alpha-oestrone series and in vitro antiproliferative properties.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 36 (1).
pp. 1931-1937.
ISSN 1475-6366
(2021)
Kiss Anita; Jójárt Rebeka; Mernyák Erzsébet; Bartha Sándor; Minorics Renáta; Zupkó István; Schneider Gyula:
Novel preparation of substituted oxazolines condensed to d-ring of estrane skeleton and characterization of their antiproliferative properties.
STEROIDS, 176.
Terjedelem: 6 p-Azonosító: 108911.
ISSN 0039-128X
(2021)
Jójárt Rebeka; Senobar Tahaei Seyyed Ashkan; Trungel-Nagy Péter; Kele Zoltán; Minorics Renáta; Paragi Gábor; Zupkó István; Mernyák Erzsébet:
Synthesis and evaluation of anticancer activities of 2- or 4-substituted 3-(N-benzyltriazolylmethyl)-13α-oestrone derivatives.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 36 (1).
pp. 58-67.
ISSN 1475-6366
(2021)
Gyovai András; Minorics Renáta; Kiss Anita; Mernyák Erzsébet; Schneider Gyula; Szekeres András; Kerekes Erika Beáta; Ocsovszki Imre; Zupkó István:
Antiproliferative properties of newly synthesized 19-nortestosterone analogs without substantial androgenic activity.
FRONTIERS IN PHARMACOLOGY, 9.
Terjedelem: 11 p.-Azonosító: 825.
ISSN 1663-9812
(2018)
Minorics Renáta; Zupkó István:
Steroidal anticancer agents: an overview of estradiol-related compounds.
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, 18 (5).
pp. 652-666.
ISSN 1871-5206
(2018)
Froehlich Tony; Kiss Anita; Wölfling János; Mernyák Erzsébet; Kulmány Ágnes Erika; Minorics Renáta; Zupkó István; Leidenberger Maria; Friedrich Oliver; Kappes Barbara; Hahn Friedrich; Marschall Manfred; Schneider Gyula; Tsogoeva Svetlana B.:
Synthesis of Artemisinin-Estrogen Hybrids Highly Active against HCMV, P-falciparum, and Cervical and Breast Cancer.
ACS MEDICINAL CHEMISTRY LETTERS, 9 (11).
pp. 1128-1133.
ISSN 1948-5875
(2018)
Bózsity Noémi; Minorics Renáta; Szabó Johanna; Mernyák Erzsébet; Schneider Gyula; Wölfling János; Wang Hui-Chun; Wu Chin-Chung; Ocsovszki Imre; Zupkó István:
Mechanism of antiproliferative action of a new D-secoestrone-triazole derivative in cervical cancer cells and its effect on cancer cell motility.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 165.
pp. 247-257.
ISSN 0960-0760
(2017)
Oprean Camelia; Zambori Csilla; Borcan Florin; Soica Codruta; Zupkó István; Minorics Renáta; Bojin Florina; Ambrus Rita; Muntean Delia; Danciu Corina; Pinzaru Iulia Andreea; Dehelean Cristina; Paunescu Virgil; Tanasie Gabriela:
Anti-proliferative and antibacterial in vitro evaluation of the polyurethane nanostructures incorporating pentacyclic triterpenes.
PHARMACEUTICAL BIOLOGY, 54 (11).
pp. 2714-2722.
ISSN 1388-0209
(2016)
Baji Ádám; Gyovai András; Wölfling János; Minorics Renáta; Ocsovszki Imre; Zupkó István; Nagyné Frank Éva:
Microwave-assisted one-pot synthesis of steroid–quinoline hybrids and an evaluation of their antiproliferative activities on gynecological cancer cell lines.
RSC ADVANCES, 6 (33).
pp. 27501-27516.
ISSN 2046-2069
(2016)
Schneider Gyula; Kiss Anita; Mernyák Erzsébet; Benke Zsanett Amália; Wölfling János; Nagyné Frank Éva; Bózsity Noémi; Gyovai András; Minorics Renáta; Zupkó István:
Stereocontrolled synthesis of the four 16-hydroxymethyl-19-nortestosterone isomers and their antiproliferative activities.
STEROIDS, 105.
pp. 113-120.
ISSN 0039-128X
(2016)
Szabó Johanna; Pataki Zoltán; Wölfling János; Schneider Gyula; Bózsity Noémi; Minorics Renáta; Zupkó István; Mernyák Erzsébet:
Synthesis and biological evaluation of 13α-estrone derivatives as potential antiproliferative agents.
STEROIDS, 113.
pp. 14-21.
ISSN 0039-128X
(2016)
Szabó Johanna; Jerkovics Nóra; Schneider Gyula; Wölfling János; Bózsity Noémi; Minorics Renáta; Zupkó István; Mernyák Erzsébet:
Synthesis and in Vitro Antiproliferative Evaluation of C-13 Epimers of Triazolyl-d-Secoestrone Alcohols: The First Potent 13alpha-d-Secoestrone Derivative.
MOLECULES, 21 (5).
Terjedelem: 13 p.-Azonosító: 611.
ISSN 1420-3049
(2016)
Molnár Judit; Nagyné Frank Éva; Minorics Renáta; Kádár Zalán; Ocsovszki Imre; Schönecker Bruno; Wölfling János; Zupkó István:
A Click Approach to Novel D-Ring-Substituted 16α-Triazolylestrone Derivatives and Characterization of Their Antiproliferative Properties.
PLOS ONE, 10 (2).
Terjedelem: 27 p.-Azonosító: e0118104.
ISSN 1932-6203
(2015)
Kovács Dóra Irén; Wölfling János; Szabó Nikoletta; Szécsi Mihály; Minorics Renáta; Zupkó István; Nagyné Frank Éva:
Efficient access to novel androsteno-17-(1′,3′,4′)-oxadiazoles and 17<beta>-(1′,3′,4′)-thiadiazoles via N-substituted hydrazone and N,N′-disubstituted hydrazine intermediates, and their pharmacological evaluation in vitro.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 98.
pp. 13-22.
ISSN 0223-5234
(2015)
Mótyán Gergő; Zupkó István; Minorics Renáta; Schneider Gyula; Wölfling János; Nagyné Frank Éva:
Lewis acid-induced intramolecular access to novel steroidal ring D-condensed arylpyrazolines exerting in vitro cell-growth-inhibitory effects.
MOLECULAR DIVERSITY, 19.
pp. 511-527.
ISSN 1381-1991
(2015)
Huber Imre; Zupkó István; Kovács Ida Jusztina; Minorics Renáta; Gulyás Gergely; Maász Gábor; Perjési Pál:
Synthesis and Antiproliferative Activity of Cyclic Arylidene Ketones: Direct Comparison of Monobenzylidene and Dibenzylidene Derivatives.
MONATSHEFTE FUR CHEMIE, 146 (6).
pp. 973-981.
ISSN 0026-9247
(2015)
Szabó Nikoletta; Iványi Zoltán; Szécsi Mihály; Julesz János; Mernyák Erzsébet; Huber Judit; Wölfling János; Minorics Renáta; Zupkó István; Schneider Gyula:
Synthesis of methoxycarbonylpyrazolylandrostene derivatives, and their potential inhibitory effect on androgen biosynthesis and cell proliferation.
Steroids, 98.
pp. 143-152.
ISSN 0039-128X
(2015)
Schneider Gyula; Görbe Tamás Ferenc; Mernyák Erzsébet; Wölfling János; Holczbauer Tamás; Czugler Mátyás; Sohár Pál; Minorics Renáta; Zupkó István:
Synthesis of novel 17-(5’-iodo)triazolyl-3-methoxyestrane epimers via Cu(I)-catalyzed azide-alkyne cycloadditon, and an evaluation of their cytotoxic activity in vitro.
STEROIDS, 98.
pp. 153-165.
ISSN 0039-128X
(2015)
Mernyák Erzsébet; Kovács Ida; Minorics Renáta; Sere Péter; Czégány Dóra; Sinka Izabella; Wölfling János; Schneider Gyula; Újfaludi Zsuzsanna; Boros Imre Miklós; Ocsovszki Imre; Varga Mónika; Zupkó István:
Synthesis of trans-16-triazolyl-13α-methyl-17-estradiol diastereomers and the effects of structural modifications on their in vitro antiproliferative activities.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 150.
pp. 123-134.
ISSN 0960-0760
(2015)
Minorics Renáta; Bózsity Noémi; Molnár Judit; Wölfling János; Mernyák Erzsébet; Schneider Gyula; Ocsovszki Imre; Zupkó István:
A molecular understanding of d-homoestrone-induced G2/M cell cycle arrest in HeLa human cervical carcinoma cells.
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 19 (10).
pp. 2365-2374.
ISSN 1582-1838
(2015)
Zupkó István; Molnár Judit; Réthy Borbála; Minorics Renáta; Nagyné Frank Éva; Wölfling János; Molnár József; Ocsovszki Imre; Topcu Zeki; Bitó Tamás; Puskás László:
Anticancer and multidrug resistance-reversal effects of solanidine analogs synthetized from pregnadienolone acetate.
MOLECULES, 19 (2).
pp. 2061-2076.
ISSN 1420-3049
(2014)
Trandafirescu Cristina; Antal Diana; Soica Codruta; Zupkó István; Minorics Renáta; Ambrus Rita; Borcan Florin; Oprean Camelia; Danciu Corina; Avram Ştefana; Dehelean Cristina; Nita Simona; Vlaia Lavinia:
Cyclodextrin Complexes of Oleanolic and Ursolic Acid: Physico-chemical and biological preliminary evaluation.
REVISTA DE CHIMIE, 65 (10).
pp. 1163-1167.
ISSN 0034-7752
(2014)
Mernyák Erzsébet; Szabó Johanna; Bacsa Ildikó; Huber Judit; Schneider Gyula; Minorics Renáta; Bózsity Noémi; Zupkó István; Varga Mónika; Bikádi Zsolt; Hazai Eszter; Wölfling János:
Syntheses and Antiproliferative Effects of D-homo- and D-secoestrones.
STEROIDS, 87.
pp. 128-136.
ISSN 0039-128X
(2014)
Mernyák Erzsébet; Huber Judit; Szabó Johanna; Schneider Gyula; Hetényi Anasztázia; Márk László; Maász Gábor; Berényi Ágnes; Kovács Ida Jusztina; Minorics Renáta; Zupkó István; Wölfling János:
Cycloaddition of Steroidal Cyclic Nitrones to C=N Dipolarophiles: Stereoselective Synthesis and Antiproliferative Effects of Oxadiazolidinones in the Estrone Series.
STEROIDS, 78 (10).
pp. 1021-1028.
ISSN 0039-128X
(2013)
Minorics Renáta; Bózsity Noémi; Wölfling János; Mernyák Erzsébet; Schneider Gyula; Márki Árpád; Falkay György; Ocsovszki Imre; Zupkó István:
Antiproliferative effect of normal and 13-epi-d-homoestrone and their 3-methyl ethers on human reproductive cancer cell lines.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 132.
pp. 168-175.
ISSN 0960-0760
(2012)
Ahmed Aimun Abdelgaffar Elhassan; Márki Árpád; Gáspár Róbert; Vasas Andrea; Mudawi Mahmoud Mudawi Eltahir; Jójárt Balázs; Minorics Renáta; Hohmann Judit; Falkay György:
In silico and in vitro pharmacological investigations of a natural alkaloid.
Medicinal Chemistry Research, 21 (12).
pp. 4100-4107.
ISSN 1054-2523
(2012)
Gáspár Róbert; Gál Adrienn; Gálik Márta; Ducza Eszter; Minorics Renáta; Klukovits Anna; Falkay György:
Different roles of alpha(2)-adrenoceptor subtypes in non-pregnant and late-pregnant uterine contractility in vitro in the rat.
NEUROCHEMISTRY INTERNATIONAL, 51 (5).
pp. 311-318.
ISSN 0197-0186
(2007)