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Pósa Vivien; Stefanelli Alessia; Nunes Julia H. Bormio; Hager Sonja; Mathuber Marlene; May Nóra Veronika; Berger Walter; Keppler Bernhard K.; Kowol Christian R.; Enyedy Éva Anna; Heffeter Petra:
Thiosemicarbazone Derivatives Developed to Overcome COTI-2 Resistance.
CANCERS, 14 (18).
Terjedelem: 27 p.-Azonosító: 4455.
ISSN 2072-6694
(2022)
Bormio Nunes Julia H.; Hager Sonja; Mathuber Marlene; Pósa Vivien; Roller Alexander; Enyedy Éva Anna; Stefanelli Alessia; Berger Walter; Keppler Bernhard K.; Heffeter Petra; Kowol Christian R.:
Cancer Cell Resistance Against the Clinically Investigated Thiosemicarbazone COTI-2 Is Based on Formation of Intracellular Copper Complex Glutathione Adducts and ABCC1-Mediated Efflux.
JOURNAL OF MEDICINAL CHEMISTRY, 63.
pp. 13719-13732.
ISSN 0022-2623
(2020)
Kallus Sebastian; Uhlik Lukas; van Schoonhoven Sushilla; Pelivan Karla; Berger Walter; Enyedy Éva Anna; Hofmann Thilo; Heffeter Petra; Kowol Christian R.; Keppler Bernhard K.:
Synthesis and biological evaluation of biotin-conjugated anticancer thiosemicarbazones and their iron(III) and copper(II) complexes.
JOURNAL OF INORGANIC BIOCHEMISTRY, 190.
pp. 85-97.
ISSN 0162-0134
(2019)
Kowol Christian R.; Walter Miklós; Pfaff Sarah; Hager Sonja; Kallus Sebastian; Pelivan Karla; Kubanik Mario; Enyedy Éva Anna; Berger Walter; Heffeter Petra; Keppler Bernhard K.:
Impact of stepwise NH2-methylation of Triapine on the physico-chemical properties, anticancer activity and resistance circumvention.
JOURNAL OF MEDICINAL CHEMISTRY, 59 (14).
pp. 6739-6752.
ISSN 0022-2623
(2016)
Martins Ana; Sipos Péter; Dér Katalin; Csábi József; Miklos Walter; Berger Walter; Zalatnai Attila; Amaral Leonard; Molnár József; Szabó-Révész Piroska; Hunyadi Attila:
Ecdysteroids sensitize MDR and non-MDR cancer cell lines to doxorubicin, paclitaxel, and vincristine but tend to protect them from cisplatin.
BioMed Research International, 2015.
Terjedelem: 8 p.-Azonosító: 895360.
ISSN 2314-6133
(2015)
Trondl Robert; Flocke Lea S.; Kowol Christian R.; Heffeter Petra; Jungwirth Ute; Mair Georg E.; Steinborn Ralf; Enyedy Éva Anna; Jakupec Michael A.; Berger Walter; Keppler Bernhard K.:
Triapine and a more potent dimethyl derivative induce ER stress in cancer cells.
MOLECULAR PHARMACOLOGY, 85 (3).
pp. 451-459.
ISSN 0026-895X
(2014)
Pichler Verena; Mayr Josef; Heffeter Petra; Dömötör Orsolya; Enyedy Éva Anna; Hermann Gerrit; Groza Diana; Köllensperger Gunda; Galanksi Markus; Berger Walter; Keppler Bernhard K.; Kowol Christian R.:
Maleimide-functionalised platinum(IV) complexes as synthetic platform for targeted drug delivery.
CHEMICAL COMMUNICATIONS, 49 (22).
pp. 2249-2251.
ISSN 1359-7345
(2013)