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Kovács Dóra Irén; Wölfling János; Szabó Nikoletta; Szécsi Mihály; Schelz Zsuzsanna; Zupkó István; Nagyné Frank Éva:
Synthesis of novel 17-(4′-formyl)pyrazolylandrosta-5,16-dienes and their derivatives as potent 17α-hydroxylase/C17,20-lyase inhibitors or antiproliferative agents depending on the substitution pattern of the heteroring.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 120.
pp. 284-295.
ISSN 0223-5234
(2016)
Kovács Dóra Irén; Wölfling János; Szabó Nikoletta; Szécsi Mihály; Minorics Renáta; Zupkó István; Nagyné Frank Éva:
Efficient access to novel androsteno-17-(1′,3′,4′)-oxadiazoles and 17<beta>-(1′,3′,4′)-thiadiazoles via N-substituted hydrazone and N,N′-disubstituted hydrazine intermediates, and their pharmacological evaluation in vitro.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 98.
pp. 13-22.
ISSN 0223-5234
(2015)
Nagyné Frank Éva; Kovács Dóra Irén; Schneider Gyula; Wölfling János; Bartók Tibor; Zupkó István:
Synthesis of novel steroidal 16-spiroisoxazolines by 1,3-dipolar cycloaddition, and an evaluation of their antiproliferative activities in vitro.
MOLECULAR DIVERSITY, 18 (3).
pp. 521-534.
ISSN 1381-1991
(2014)