Vissza |
Peřina Miroslav; Kiss Márton Attila; Mótyán Gergő; Szczyrbová Eva; Eliáš Martin; Student jr Vladimír; Kurfürstova Daniela; Kovalova Marketa; Mada Lukáš; Bouchal Jan; Nagyné Frank Éva; Jorda Radek:
A-ring-fused pyrazoles of dihydrotestosterone targeting prostate cancer cells via the downregulation of the androgen receptor.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 249.
ISSN 0223-5234
(2023)
Kiss Márton Attila; Peřina Miroslav; Bereczki Laura; Baji Ádám; Bělíček Jakub; Jorda Radek; Nagyné Frank Éva:
Dihydrotestosterone-based A-ring-fused pyridines: microwave-assisted synthesis and biological evaluation in prostate cancer cells compared to structurally related quinolines.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 231.
ISSN 0960-0760
(2023)
Peřina Miroslav; Kiss Anita; Mernyák Erzsébet; Mada Lukáš; Schneider Gyula; Jorda Radek:
Synthesis of hydrocortisone esters targeting androgen and glucocorticoid receptors in prostate cancer in vitro.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 229.
ISSN 0960-0760
(2023)
Kiss Márton Attila; Miroslav Peřina; Václav Bazgier; May Nóra V.; Baji Ádám; Jorda Radek; Nagyné Frank Éva:
Synthesis of dihydrotestosterone derivatives modified in the A-ring with (hetero)arylidene, pyrazolo[1,5-a]pyrimidine and triazolo[1,5-a]pyrimidine moieties and their targeting of the androgen receptor in prostate cancer.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 211.
Terjedelem: 17 p-Azonosító: 105904.
ISSN 0960-0760
(2021)