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Bormio Nunes, Julia H., Hager, Sonja, Mathuber, Marlene, Pósa, Vivien, Roller, Alexander, Enyedy, Éva Anna, Stefanelli, Alessia, Berger, Walter, Keppler, Bernhard K., Heffeter, Petra, Kowol, Christian R.:
Cancer Cell Resistance Against the Clinically Investigated Thiosemicarbazone COTI-2 Is Based on Formation of Intracellular Copper Complex Glutathione Adducts and ABCC1-Mediated Efflux.
JOURNAL OF MEDICINAL CHEMISTRY, 63.
pp. 13719-13732.
ISSN 0022-2623
(2020)
Enyedy, Éva Anna, May, Nóra Veronika, Pape, Veronika, Heffeter, Petra, Szakács, Gergely, Keppler, Bernhard K., Kowol, Christian R.:
Complex formation and cytotoxicity of Triapine derivatives: a comparative solution study on the effect of the chalcogen atom and NH-methylation.
DALTON TRANSACTIONS, 49.
pp. 16887-16902.
ISSN 1477-9226
(2020)
Hager, Sonja, Pape, Veronika, Pósa, Vivien, Montsch, Bianca, Uhlik, Lukas, Szakács, Gergely, Tóth, Szilárd, Jabronka, Nikolett, Keppler, Bernhard K., Kowol, Christian R., Enyedy, Éva Anna, Heffeter, Petra:
High copper complex stability and slow reduction kinetics as key parameters for improved activity, paraptosis induction and impact on drug-resistant cells of anticancer thiosemicarbazones.
ANTIOXIDANTS & REDOX SIGNALING, 33 (6).
pp. 395-414.
ISSN 1523-0864
(2020)
Mathuber, Marlene, Schueffl, Hemma, Dömötör, Orsolya, Karnthaler, Claudia, Enyedy, Éva Anna, Heffeter, Petra, Kowol, Christian R.:
Improving the Stability of EGFR Inhibitor Cobalt(III) Prodrugs.
INORGANIC CHEMISTRY, 59 (23).
pp. 17794-17810.
ISSN 0020-1669
(2020)
Heffeter, Petra, Pape, Veronika, Enyedy, Éva Anna, Keppler, Bernhard K., Szakács, Gergely, Kowol, Christian R.:
Anticancer thiosemicarbazones: chemical properties, interaction with iron metabolism, and resistance development.
ANTIOXIDANTS & REDOX SIGNALING, 30 (8).
pp. 1062-1082.
ISSN 1523-0864
(2019)
Kallus, Sebastian, Uhlik, Lukas, van Schoonhoven, Sushilla, Pelivan, Karla, Berger, Walter, Enyedy, Éva Anna, Hofmann, Thilo, Heffeter, Petra, Kowol, Christian R., Keppler, Bernhard K.:
Synthesis and biological evaluation of biotin-conjugated anticancer thiosemicarbazones and their iron(III) and copper(II) complexes.
JOURNAL OF INORGANIC BIOCHEMISTRY, 190.
pp. 85-97.
ISSN 0162-0134
(2019)
Kowol, Christian R., Walter, Miklós, Pfaff, Sarah, Hager, Sonja, Kallus, Sebastian, Pelivan, Karla, Kubanik, Mario, Enyedy, Éva Anna, Berger, Walter, Heffeter, Petra, Keppler, Bernhard K.:
Impact of stepwise NH2-methylation of Triapine on the physico-chemical properties, anticancer activity and resistance circumvention.
JOURNAL OF MEDICINAL CHEMISTRY, 59 (14).
pp. 6739-6752.
ISSN 0022-2623
(2016)
Kowol, Christian R., Nagy, Nóra Veronika, Jakusch, Tamás, Roller, Alexander, Heffeter, Petra, Keppler, Bernhard K., Enyedy, Éva Anna:
Vanadium(IV/V) complexes of Triapine and related thiosemicarbazones: synthesis, solution equilibrium and bioactivity.
JOURNAL OF INORGANIC BIOCHEMISTRY, 152 (SI).
pp. 62-73.
ISSN 0162-0134
(2015)
Trondl, Robert, Flocke, Lea S., Kowol, Christian R., Heffeter, Petra, Jungwirth, Ute, Mair, Georg E., Steinborn, Ralf, Enyedy, Éva Anna, Jakupec, Michael A., Berger, Walter, Keppler, Bernhard K.:
Triapine and a more potent dimethyl derivative induce ER stress in cancer cells.
MOLECULAR PHARMACOLOGY, 85 (3).
pp. 451-459.
ISSN 0026-895X
(2014)
Pichler, Verena, Mayr, Josef, Heffeter, Petra, Dömötör, Orsolya, Enyedy, Éva Anna, Hermann, Gerrit, Groza, Diana, Köllensperger, Gunda, Galanksi, Markus, Berger, Walter, Keppler, Bernhard K., Kowol, Christian R.:
Maleimide-functionalised platinum(IV) complexes as synthetic platform for targeted drug delivery.
CHEMICAL COMMUNICATIONS, 49 (22).
pp. 2249-2251.
ISSN 1359-7345
(2013)