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Pósa Vivien; Stefanelli Alessia; Nunes Julia H. Bormio; Hager Sonja; Mathuber Marlene; May Nóra Veronika; Berger Walter; Keppler Bernhard K.; Kowol Christian R.; Enyedy Éva Anna; Heffeter Petra:
Thiosemicarbazone Derivatives Developed to Overcome COTI-2 Resistance.
CANCERS, 14 (18).
Terjedelem: 27 p.-Azonosító: 4455.
ISSN 2072-6694
(2022)
Bormio Nunes Julia H.; Hager Sonja; Mathuber Marlene; Pósa Vivien; Roller Alexander; Enyedy Éva Anna; Stefanelli Alessia; Berger Walter; Keppler Bernhard K.; Heffeter Petra; Kowol Christian R.:
Cancer Cell Resistance Against the Clinically Investigated Thiosemicarbazone COTI-2 Is Based on Formation of Intracellular Copper Complex Glutathione Adducts and ABCC1-Mediated Efflux.
JOURNAL OF MEDICINAL CHEMISTRY, 63.
pp. 13719-13732.
ISSN 0022-2623
(2020)
Hager Sonja; Pape Veronika; Pósa Vivien; Montsch Bianca; Uhlik Lukas; Szakács Gergely; Tóth Szilárd; Jabronka Nikolett; Keppler Bernhard K.; Kowol Christian R.; Enyedy Éva Anna; Heffeter Petra:
High copper complex stability and slow reduction kinetics as key parameters for improved activity, paraptosis induction and impact on drug-resistant cells of anticancer thiosemicarbazones.
ANTIOXIDANTS & REDOX SIGNALING, 33 (6).
pp. 395-414.
ISSN 1523-0864
(2020)
Kowol Christian R.; Walter Miklós; Pfaff Sarah; Hager Sonja; Kallus Sebastian; Pelivan Karla; Kubanik Mario; Enyedy Éva Anna; Berger Walter; Heffeter Petra; Keppler Bernhard K.:
Impact of stepwise NH2-methylation of Triapine on the physico-chemical properties, anticancer activity and resistance circumvention.
JOURNAL OF MEDICINAL CHEMISTRY, 59 (14).
pp. 6739-6752.
ISSN 0022-2623
(2016)