Vissza |
Kiss Márton Attila; Peřina Miroslav; Bereczki Laura; Baji Ádám; Bělíček Jakub; Jorda Radek; Nagyné Frank Éva:
Dihydrotestosterone-based A-ring-fused pyridines: microwave-assisted synthesis and biological evaluation in prostate cancer cells compared to structurally related quinolines.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 231.
ISSN 0960-0760
(2023)
Nagy Ferenc István; Adamecz Dóra Izabella; Baji Ádám; Kiricsi Ágnes; Huliák Ildikó; Rónavári Andrea; Kónya Zoltán; Nagyné Frank Éva; Gopisetty Mohana Krishna; Csontné Kiricsi Mónika:
Semi-Synthetic Dihydrotestosterone Derivatives Modulate Inherent Multidrug Resistance and Sensitize Colon Cancer Cells to Chemotherapy.
PHARMACEUTICS, 15 (2).
ISSN 1999-4923
(2023)
Gopisetty Mohana Krishna; Adamecz Dóra Izabella; Nagy Ferenc István; Baji Ádám; Lathira Vasiliki; Szabó Márton Richárd; Gáspár Renáta; Csont Tamás Bálint; Nagyné Frank Éva; Csontné Kiricsi Mónika:
Androstano-arylpyrimidines : novel small molecule inhibitors of MDR1 for sensitizing multidrug-resistant breast cancer cells.
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 156.
Terjedelem: 11 p-Azonosító: 105587.
ISSN 0928-0987
(2021)
Kiss Márton Attila; Miroslav Peřina; Václav Bazgier; May Nóra V.; Baji Ádám; Jorda Radek; Nagyné Frank Éva:
Synthesis of dihydrotestosterone derivatives modified in the A-ring with (hetero)arylidene, pyrazolo[1,5-a]pyrimidine and triazolo[1,5-a]pyrimidine moieties and their targeting of the androgen receptor in prostate cancer.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 211.
Terjedelem: 17 p-Azonosító: 105904.
ISSN 0960-0760
(2021)
Mótyán Gergő; Baji Ádám; Marć Małgorzata Anna; Gopisetty Mohana Krishna; Adamecz Dóra Izabella; Csontné Kiricsi Mónika; Enyedy Éva Anna; Nagyné Frank Éva:
Microwave-Assisted Synthesis, Proton Dissociation Processes, and Anticancer Evaluation of Novel D-Ring-Fused Steroidal 5-Amino-1-Arylpyrazoles.
APPLIED SCIENCES-BASEL, 10 (1).
Azonosító: 229-Terjedelem: 13 p.
ISSN 2076-3417
(2020)
Baji Ádám; Kovács Ferenc; Mótyán Gergő; Schneider Gyula; Wölfling János; Sinka Izabella; Zupkó István; Ocsovszki Imre; Nagyné Frank Éva:
Investigation of pH and substituent effects on the distribution ratio of novel steroidal ring D- and A-fused arylpyrazole regioisomers and evaluation of their cell-growth inhibitory effects in vitro.
STEROIDS, 126.
pp. 35-49.
ISSN 0039-128X
(2017)
Baji Ádám; Kiss Tamás; Wölfling János; Kovács Dávid; Igaz Nóra; Gopisetty Mohana Krishna; Kiricsi Mónika; Frank Éva:
Multicomponent access to androstano-arylpyrimidines under microwave conditions and evaluation of their anti-cancer activity in vitro.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 172.
pp. 79-88.
ISSN 0960-0760
(2017)
Baji Ádám; Gyovai András; Wölfling János; Minorics Renáta; Ocsovszki Imre; Zupkó István; Nagyné Frank Éva:
Microwave-assisted one-pot synthesis of steroid–quinoline hybrids and an evaluation of their antiproliferative activities on gynecological cancer cell lines.
RSC ADVANCES, 6 (33).
pp. 27501-27516.
ISSN 2046-2069
(2016)
Mótyán Gergő; Baji Ádám; Zupkó István; Nagyné Frank Éva:
Regio- and stereoselective synthesis of pregnane-fused isoxazolines by nitril-oxide/alkene 1,3-dipolar cycloaddition and an evaluation of their cell-growth inhibitory effect in vitro.
JOURNAL OF MOLECULAR STRUCTURE, 1110.
pp. 143-149.
ISSN 0022-2860
(2016)