TY - JOUR ID - publicatio31967 AV - restricted A1 - Kóbor Jen? A1 - Lázár János A1 - Fülöp Ferenc A1 - Bernáth Gábor Y1 - 1994/// EP - 828 VL - 31 SN - 0022-152X JF - JOURNAL OF HETEROCYCLIC CHEMISTRY IS - 4 TI - Saturated heterocycles. Part 209. Synthesis of 1?cyclohexyl?substituted isoquinoline derivatives N2 - In contrast with earlier literature data [7], both acrylic esters and acrylonitrile underwent Michael addition to 1-methyl-3,4-dihydroisoquinolines 14 to yield the diesters 5-9 or the dinitrile 10, respectively. Compounds S-10 were converted by Claisen condensation to 1-[(3'-methoxycarbonyl- or 1-[(3'-ethoxycarbonyl-4'-oxo)-1-cyclohexyl]-3,4-dihydroisoquinoline derivatives 11-16. Several derivatives of 12 were prepared. The new compounds possess various pharmacological actions. UR - https://doi.org/10.1002/jhet.5570310423 SP - 825 ER -